Search Results - "Bury, Paul"

Genome-wide association mapping to candidate polymorphism resolution in the unsequenced barley genome by Cockram, James, White, Jon, Zuluaga, Diana L., Smith, David, Comadran, Jordi, Macaulay, Malcolm, Luo, Zewei, Kearsey, Mike J., Werner, Peter, Harrap, David, Tapsell, Chris, Liu, Hui, Hedley, Peter E., Stein, Nils, Schulte, Daniela, Steuernagel, Burkhard, Marshall, David F., Thomas, William T. B., Ramsay, Luke, Mackay, Ian, Balding, David J., Waugh, Robbie, O'Sullivan, Donal M., Doebley, John

“…Although commonplace in human disease genetics, genome-wide association (GWA) studies have only relatively recently been applied to plants. Using 32 phenotypes…”
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Map-based cloning of the fertility restoration locus Rfm1 in cultivated barley (Hordeum vulgare) by Rizzolatti, Carine, Bury, Paul, Tatara, Edouard, Pin, Pierre A., Rodde, Nathalie, Bergès, Hélène, Budar, Françoise, Mireau, Hakim, Gielen, Jan J. L.

“…Hybridization technology has proven valuable in enhancing yields in many crops, but was only recently adopted in the small grain cereals. Hybrid varieties in…”
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Novel Tricyclic-α-alkyloxyphenylpropionic Acids:  Dual PPARα/γ Agonists with Hypolipidemic and Antidiabetic Activity by Sauerberg, Per, Pettersson, Ingrid, Jeppesen, Lone, Bury, Paul S, Mogensen, John P, Wassermann, Karsten, Brand, Christian L, Sturis, Jeppe, Wöldike, Helle F, Fleckner, Jan, Andersen, Anne-Sofie T, Mortensen, Steen B, Svensson, L. Anders, Rasmussen, Hanne B, Lehmann, Søren V, Polivka, Zdenek, Sindelar, Karel, Panajotova, Vladimira, Ynddal, Lars, Wulff, Erik M

“…Synthesis and structure−activity relationships of tricyclic α-ethoxy-phenylpropionic acid derivatives guided by in vitro PPARα and PPARγ transactivation data…”
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Design of potent PPARα agonists by Sauerberg, Per, Mogensen, John P., Jeppesen, Lone, Bury, Paul S., Fleckner, Jan, Olsen, Grith S., Jeppesen, Claus B., Wulff, Erik M., Pihera, Pavel, Havranek, Miroslav, Polivka, Zdenek, Pettersson, Ingrid

“…Computational analysis of the ligand binding pocket of the three PPAR receptor subtypes was utilized in the design of potent PPARα agonists. Optimum PPARα…”
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Selective estrogen receptor modulator effects in the rat brain by Zhou, Wenxia, Koldzic-Zivanovic, Nina, Clarke, Charlotte H, de Beun, René, Wassermann, Karsten, Bury, Paul S, Cunningham, Kathryn A, Thomas, Mary L

“…The effects in the brain of selective estrogen receptor modulators (SERMs) such as tamoxifen and raloxifene have not yet been fully elucidated. Based upon the…”
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Large Dimeric Ligands with Favorable Pharmacokinetic Properties and Peroxisome Proliferator-Activated Receptor Agonist Activity in Vitro and in Vivo by Sauerberg, Per, Bury, Paul S, Mogensen, John P, Deussen, Heinz-Josef, Pettersson, Ingrid, Fleckner, Jan, Nehlin, Jan, Frederiksen, Klaus S, Albrektsen, Tatjana, Din, Nanni, Svensson, L. Anders, Ynddal, Lars, Wulff, Erik M, Jeppesen, Lone

“…Two potent nonselective, but PPARα-preferring, PPAR agonists 5 and 6 were designed and synthesized in high yields. The concept of dimeric ligands in…”
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Design and synthesis of novel PPARα/γ/δ triple activators using a known PPARα/γ dual activator as structural template by Mogensen, John P, Jeppesen, Lone, Bury, Paul S, Pettersson, Ingrid, Fleckner, Jan, Nehlin, Jan, Frederiksen, Klaus S, Albrektsen, Tatjana, Din, Nanni, Mortensen, Steen B, Svensson, L.Anders, Wassermann, Karsten, Wulff, Erik M, Ynddal, Lars, Sauerberg, Per

“…Using a known dual PPARα/γ activator ( 5) as a structural template, SAR evaluations led to the identification of triple PPARα/γ/δ activators ( 18– 20) with…”
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Photo-removable protecting groups for in situ DNA microarray synthesis by Afroz, Farhana, Barone, Anthony D, Bury, Paul A, Chen, Chuan, Cuppoletti, Andrea, Kuimelis, Robert G, Li, Handong, McGall, Glenn H

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Synthesis and estrogen receptor binding affinities of novel pyrrolo[2,1,5- cd]indolizine derivatives by Jørgensen, Anker Steen, Jacobsen, Poul, Christiansen, Lise Brown, Bury, Paul S., Kanstrup, Anders, Thorpe, Susan M., Nærum, Lars, Wassermann, Karsten

“…A series of pyrrolo[2,1,5- cd]indolizine derivatives has been synthesized and evaluated as ligands for the estrogen receptor. Properly substituted mono- and…”
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Synthesis and pharmacological evaluation of novel cis-3,4-Diaryl-hydroxychromanes as high affinity partial agonists for the estrogen receptor by Bury, Paul S., Christiansen, Lise B., Jacobsen, Poul, Jørgensen, Anker S., Kanstrup, Anders, Nærum, Lars, Bain, Steven, Fledelius, Christian, Gissel, Birgitte, Hansen, Birgit S., Korsgaard, Niels, Thorpe, Susan M., Wassermann, Karsten

“…The syntheses and in vitro pharmacological evaluation of a number of cis-3,4-diaryl-hydroxy-chromanes are reported, along with the results of a thorough in…”
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Hybrid Breeding in Barley by Mühleisen, Jonathan, Maurer, Hans Peter, Stiewe, Gunther, Bury, Paul, Reif, Jochen C.

“…ABSTRACT Barley (Hordeum vulgare L.) has been largely neglected in hybrid breeding research of autogamous cereals. The objectives of our study were (i) to…”
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Synthesis and biological evaluation of novel thio-substituted chromanes as high-affinity partial agonists for the estrogen receptor by Christiansen, Lise B, Wenckens, Martin, Bury, Paul S, Gissel, Birgitte, Hansen, Birgit S, Thorpe, Susan M, Jacobsen, Poul, Kanstrup, Anders, Jørgensen, Anker S, Nærum, Lars, Wassermann, Karsten

“…Synthesis of (±)- cis-7-hydroxy-3-phenyl-4-(4-(2-piperidinoethanethio)phenyl)chromane ( 13) and (±)-…”
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Design of potent PPARalpha agonists by Sauerberg, Per, Mogensen, John P, Jeppesen, Lone, Bury, Paul S, Fleckner, Jan, Olsen, Grith S, Jeppesen, Claus B, Wulff, Erik M, Pihera, Pavel, Havranek, Miroslav, Polivka, Zdenek, Pettersson, Ingrid

“…Computational analysis of the ligand binding pocket of the three PPAR receptor subtypes was utilized in the design of potent PPARalpha agonists. Optimum…”
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Directed ortho metalation - cross coupling connections. Remote lateral metalation - cyclization of 2-imino-2′-methyl biaryls to 9-aminophenanthrenes. A synthesis of the alkaloid piperolactam C by Benesch, Lisbeth, Bury, Paul, Guillaneux, Denis, Houldsworth, Stephen, Wang, X., Snieckus, Victor

“…2-Imino-2′-methyl biaryls, conveniently available by Suzuki cross coupling protocol, undergo lithium diethyl amide-mediated metalation - cyclization to give…”
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PHOTOLITHOGRAPHIC SYNTHESIS OF HIGH-DENSITY OLIGONUCLEOTIDE PROBE ARRAYS by Barone, Anthony D., Beecher, Jody E., Bury, Paul A., Chen, Chuan, Doede, Tina, Fidanza, Jacqueline A., McGall, Glenn H.

“…High-density DNA probe arrays provide a massively parallel approach to nucleic acid sequence analysis that is transforming gene-based biomedical research and…”
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Design and synthesis of novel PPARalpha/gamma/delta triple activators using a known PPARalpha/gamma dual activator as structural template by Mogensen, John P, Jeppesen, Lone, Bury, Paul S, Pettersson, Ingrid, Fleckner, Jan, Nehlin, Jan, Frederiksen, Klaus S, Albrektsen, Tatjana, Din, Nanni, Mortensen, Steen B, Svensson, L Anders, Wassermann, Karsten, Wulff, Erik M, Ynddal, Lars, Sauerberg, Per

“…Using a known dual PPARalpha/gamma activator (5) as a structural template, SAR evaluations led to the identification of triple PPARalpha/gamma/delta activators…”
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Novel tricyclic-alpha-alkyloxyphenylpropionic acids: dual PPARalpha/gamma agonists with hypolipidemic and antidiabetic activity by Sauerberg, Per, Pettersson, Ingrid, Jeppesen, Lone, Bury, Paul S, Mogensen, John P, Wassermann, Karsten, Brand, Christian L, Sturis, Jeppe, Wöldike, Helle F, Fleckner, Jan, Andersen, Anne-Sofie T, Mortensen, Steen B, Svensson, L Anders, Rasmussen, Hanne B, Lehmann, Søren V, Polivka, Zdenek, Sindelar, Karel, Panajotova, Vladimira, Ynddal, Lars, Wulff, Erik M

“…Synthesis and structure-activity relationships of tricyclic alpha-ethoxy-phenylpropionic acid derivatives guided by in vitro PPARalpha and PPARgamma…”
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Enzymatic resolution to (?)-ormeloxifene intermediates from their racemates using immobilizedCandida rugosa lipase by Lehmann, S ren Vig, Breinholt, Jens, Bury, Paul Stanley, Nielsen, Thomas Eiland

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Enzymatic resolution to (−)-ormeloxifene intermediates from their racemates using immobilized Candida rugosa lipase by Lehmann, Søren Vig, Breinholt, Jens, Bury, Paul Stanley, Nielsen, Thomas Eiland

“…In the synthesis of (−)‐ormeloxifene, a drug candidate recently under development, enzymatic resolution of potential intermediates can be carried out using a…”
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Drug-using mothers: social, psychological and substance use problems of women opiate users with children by Powis, Michael Gossop, Catherine Bury, Katherine Payne, Paul Griffiths, Beverly

“…The present study looks at patterns of drug use and alcohol use, social and economic circumstances, criminal involvement and health problems among a sample of…”
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