Search Results - "Bruzzese, T"

Analgesic effect of bisphosphonates in mice by Bonabello, A, Galmozzi, M.R, Bruzzese, T, Zara, G.P

“…Bisphosphonates are analogues of inorganic pyrophosphate and are inhibitors of bone resorption. Many derivatives have been developed for the treatment of…”
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In Vitro Activity of a New Polyene, SPA-S-843, against Yeasts by RIMAROLI, C, BRUZZESE, T

“…Classifications Services AAC Citing Articles Google Scholar PubMed Related Content Social Bookmarking CiteULike Delicious Digg Facebook Google+ Mendeley Reddit…”
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The use of lipid emulsions for the iv administration of a new water soluble polyene antibiotic, SPK-843 by Mozzi, G., Benelli, P., Bruzzese, T., Galmozzi, M. R., Bonabello, A.

“…Venous tolerance of a new water soluble polyene antibiotic, SPK-843, in 5% glucose solution for infusion is low in laboratory animals. The use of Intralipid…”
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Effects of mepartricin on estradiol and testosterone serum levels and on prostatic estrogen, androgen and adrenergic receptor concentrations in adult rats by Re, G., Badino, P., Odore, R., Vigo, D., Bonabello, A., Rabino, S., Capello, F., Bruzzese, T.

“…The effects induced by oral administration of 0, 5 and 20 mg of meparticin kg−1of body weight for 28 days (group 1, 2 and 3, respectively) upon prostatic…”
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Amide derivatives of partricin A with potent antifungal activity by Bruzzese, T, Rimaroli, C, Bonabello, A, Ferrari, E, Signorini, M

“…A series of partricin A amides were synthesized using the active ester method by reaction with several amines on the carboxy group and then with some acids on…”
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Anticandidal activity of SPA-S-843, a new polyenic drug by STRIPPOLI, V, D'AURIA, F. D, SIMONETTI, G, BRUZZESE, T, SIMONETTI, N

“…The activity of a new, soluble and stable polyene (SPA-S-843) against Candida albicans was assessed by contact and culture tests and by inhibition of germ-tube…”
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Pharmacokinetics in rats of n-dimethylaminoacetyl-partricin a 2-dimethylaminoethylamide diascorbate (spk-843) by Bruzzese, T, Galmozzi, M R, Buffa, G, Sala, P, Bonabello, A

“…Single- and multiple-administration trials in rats were performed in this study to assess the serum and tissue concentrations of SPK-843…”
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Pharmacokinetics of a new derivative of partricin A (SPA-S-753) in rodents by Galmozzi, M R, Bruzzese, T, Buffa, G, Bonabello, A

“…Pharmacokinetics of a new semisynthetic polyene antibiotic (N-dimethylaminoacetyl-partricin A 2-dimethylaminoethylamide) in the form of its diaspartate salt…”
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Comparative pharmacokinetics of three preparations of the new antifungal SPK-843 by Bruzzese, T, Galmozzi, M R, Ferrari, V M, Sala, P, Bonabello, A

“…The pharmacokinetics and tissue distribution of three preparations of SPK-843 (N-dimethylaminoacetyl-partricin A 2-dimethylaminoethylamide diascorbate), a new…”
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Comparative anti-gonococcal activity of S-565, a new rifamycin by Hamilton-Miller, J.M.T., Bruzzese, T., Nonis, A., Shah, S.

“…The in vitro activity of S-565, a semi-synthetic rifamycin chemically related to rifampicin but with a longer half-life, has been compared with that of…”
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Phase I pharmacokinetic study of a new 3-azinomethyl-rifamycin (rifametane) as compared to rifampicin by Potkar, C, Gogtay, N, Gokhale, P, Kshirsagar, N A, Ajay, S, Cooverji, N D, Bruzzese, T

“…An open randomized cross-over study was conducted in 8 healthy male volunteers to study the pharmacokinetic pattern and the safety of a 300-mg single oral dose…”
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In vivo and in vitro antifungal activity of the polyene derivative SPA-S-753 against encapsulated form of Cryptococcus neoformans by STRIPPOLI, V, D'AURIA, F. D, SIMONETTI, N, BASTI, D, BRUZZESE, T

“…The in vitro and in vivo activity of SPA-S-753 (N-dimethylaminoacetyl-partricin A 2-dimethylaminoethylamide diaspartate), a new water soluble polyene, was…”
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Pharmacokinetic profile of a new 3-azinomethyl rifamycin (SPA-S-565) in volunteers as compared with conventional rifampicin by Kelkar, M S, Saraf, A P, Bakhle, D S, Nazare, V, Ajay, S, Hegde, S, Lal, H M, Cooverji, N D, Bruzzese, T

“…The pharmacokinetics and tolerance of a single oral dose (150 mg) of a new 3-azinomethyl rifamycin (SPA-S-565, USAN rifametane) was compared with 150 mg of…”
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Synthesis and biological properties of alkyl esters of polyene antibiotics by Bruzzese, T, Cambieri, M, Recusani, F

“…Several new alkyl esters of polyene antibiotics were prepared by an improved general procedure, and their toxicity and microbiological activity were tested…”
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Relationship between acute toxicity in mice and polymorphic forms of polyene antibiotics by Ghielmetti, G, Bruzzese, T, Bianchi, C, Recusani, F

“…Marked differences in LD50 values were found between various batches of polyene antibiotics (mepartricin and nystatin) after intraperitoneal administration in…”
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Guanidinated derivatives of lysozyme by Bruzzese, T, Cambieri, M

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Binding of Mepartricin to Sex Hormones, a Key Factor of its Activity on Benign Prostatic Hyperplasia by Barone, Domenico, Peroglio, Flavio, Toso, Emiliano, Bruzzese, Tiberio

“…Summary Androgens and estrogens, mainly testosterone (TES) and dihydrotestosterone (DHT) and 17ß-estradiol (EST), are widely recognized to regulate the…”
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The antibacterial activity of a new 3-azinomethyl-rifamycin by Strippoli, V, Bruzzese, T, Galli, R, Simonetti, N, Tronci, N

“…The new 3-azinomethyl-rifamycin, SPA-S-565, was shown to exert an effective antibacterial activity in vitro comparable to that of rifampicin. In fact, the…”
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Complex partial status epilepticus simulating an ischemic insult: case report by Musolino, R, Marabello, L, De Domenico, P, Labate, C, Bruzzese, T, Galatioto, S, Gallitto, G

“…A patient presenting complex partial status epilepticus (CPSE) had a clinical history and neurological picture on admission that mimicked a cerebrovascular…”
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Pharmacokinetics and tissue distribution of a new partricin A derivative (N-dimethylaminoacetyl-partricin A 2-dimethylaminoethylamide diaspartate) in mice by Rimaroli, Claudio, Bonabello, Angelo, Sala, Patrizio, Bruzzese, Tiberio

“…A single-dose trial in mice (1.25 mg/kg SPA-S-753 or 1 mg/kg amphotericin B [AmB] by intravenous route) was performed to study the pharmacokinetics, tissue…”
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