Search Results - "Brouant, P"

Structure and conformational analysis of 5,11-dibenzyldibenzo[b,f][1,5]diazocine-6,12-dione. A novel approach for new chemosensitizers by Nonnenmacher, E, Brouant, P, Mrozek, A, Karolak-Wojciechowska, J, Barbe, J

“…On the basis of structural similarities between various calcium channel antagonists (Verapamil or Diltiazem) a novel series of derivatives belonging to the…”
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2-Anilino-4,6-dimethylpyridine-3-carbonitrile, an Intermediate in the Synthesis of 5-Aminobenzo[b][1,8]naphthyridines by Mefetah, H., Giorgi, M., Brouant, P.

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Antimicrobial activity of 9-oxo and 9-thio acridines: Correlation with intercalation into DNA and effects on macromolecular biosynthesis by Crémieux, A, Chevalier, J, Sharples, D, Berny, H, Galy, A.M, Brouant, P, Galy, J.P, Barbe, J

“…The antimicrobial activity of several new 9-acridinones and 9-thioalkylacridines towards Escherichia coli, Staphylococcus aureus, Mycobacterium smegmatis and…”
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Alkylaminoquinolines inhibit the bacterial antibiotic efflux pump in multidrug-resistant clinical isolates by Malléa, Monique, Mahamoud, Abdallah, Chevalier, Jacqueline, Alibert-Franco, Sandrine, Brouant, Pierre, Barbe, Jacques, Pagès, Jean-Marie

“…Over the last decade, MDR (multidrug resistance) has increased worldwide in microbial pathogens by efflux mechanisms, leading to treatment failures in human…”
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Modified electrodes with new phenothiazine derivatives for electrocatyltic oxidation of NADH by Dicu, Delia, Muresan, Liana, Popescu, Ionel Catalin, Cristea, Castelia, Silberg, Ioan Alexandru, Brouant, Pierre

“…Phenothiazine derivatives containing two linearly condensed phenothiazine moieties, 16 H,18 H-dibenzo[c,l]-7,9-dithia-16,18-diazapentacene (I), dibenzo[c,l]-16…”
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Benzo[b]-1,8-naphthyridine derivatives: synthesis and reversal activity on multidrug resistance by Misbahi, Houria, Brouant, Pierre, Hevér, Aniko, Molnár, Anna Maria, Wolfard, Krysztina, Spengler, Grabriela, Mefetah, Hafid, Molnár, Joseph, Barbe, Jacques

“…A series of benzo[b]-1,8-naphthyridine derivatives branched with various side-chains and substituents were prepared with the aim of being investigated as…”
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Membrane Permeation by Multidrug-resistance-modulators and Non-modulators: Effects of Hydrophobicity and Electric Charge by CASTAING, MADELEINE, BROUANT, PIERRE, LOISEAU, ALAIN, SANTELLI-ROUVIER, CHRISTIANE, SANTELLI, MAURICE, ALIBERT-FRANCO, SANDRINE, MAHAMOUD, ABDALLAH, BARBE, JACQUES

“…This study was designed to test the hypothesis that lipophilic cationic drugs with only roughly similar structures mediate the reversal of multidrug‐resistance…”
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Effect of new thioacridine derivatives on P-gp function and on mdr1 gene expression by Hevér, A, Santelli-Rouvier, C, Brouant, P, el Khyari, S, Molnár, J, Barra, Y, Barbe, J

“…We studied the effect of thioacridine derivatives on the function of P-glycoprotein in MDR mouse T-lymphoma cell line L5178 and in MDR human leukemia cell line…”
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Synthesis of new bis(2,4-dimethyl-5-amino-benzo[b][1,8]-naphthyridines) and bis(benzo[b][1,8]naphthyridones) linked with methylene linear chain by Afloroaei, Cerasella, Dulamita, Nicu, Vlassa, Mircea, Barbe, Jacques, Brouant, Pierre

“…The preparation of novel alkyl monobridged 2,4‐dimethyl‐5‐amino‐benzo[b][1,8]naphthyiridine and benzo[b][1,8]naphthyridone derivatives by phase transfer…”
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Computer simulation of spermine-porin channel interactions by Vidal, Stéphanie, Brouant, Pierre, Chevalier, Jacqueline, Malléa, Monique, Barbe, Jacques, Pagès, Jean-Marie

“…Porin channels play a prominent role during fluoroquinolone uptake and spermine strongly alters the diffusion rate of norfloxacine. Consequently the…”
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Antimicrobial activity of 9-oxo and 9-thio acridines: correlation with interacalation into DNA and effects on macromolecular biosynthesis by Crémieux, A, Chevalier, J, Sharples, D, Berny, H, Galy, A M, Brouant, P, Galy, J P, Barbe, J

“…The antimicrobial activity of several new 9-acridinones and 9-thioalkylacridines towards Escherichia coli, Staphylococcus aureus, Mycobacterium smegmatis and…”
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Variation of the conformational background of morphinic analgesics through their radiocrystallographic study (author's transl) by Brouant, P, Soyfer, J C

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Phenylpropylamino groups of morphine analgesics plotted with a computer (author's transl) by Brouant, P, Soyfer, J C

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Inhibition of cryptosporidium parvum in vitro by 9-(alkylthio)acridine derivatives by KHALIFA, L, ROSALES, M.-J, MASCARO, C, KAROLAK-WOJCIECHOWSKA, J, BSIRI, N, BROUANT, P, BARBE, J

“…The synthesis of several acridinic thioethers is described. Compounds prepared were tested in vitro as potential drugs against the opportunistic infection…”
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Identification and analysis of commercial isoborneol and borneol by gas phase chromatography and proton N.M.R by Brouant, P, Reboul, J P, Cristau, B

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