Search Results - "Brel, Valery K."

Design of Conjugates Based on Sesquiterpene Lactones with Polyalkoxybenzenes by "Click" Chemistry to Create Potential Anticancer Agents by Neganova, Margarita E, Smirnova, Ekaterina V, Sharova, Elena V, Artyushin, Oleg I, Aleksandrova, Yulia R, Yandulova, Ekaterina Yu, Nikolaeva, Natalia S, Brel, Valery K

“…Using the methodology of "click" chemistry, a singular method has been developed for the synthesis of unique conjugates based on sesquiterpene lactones:…”
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Synthesis and biological testing of 3,5-bis(arylidene)-4-piperidone conjugates with 2,5-dihydro-5H-1,2-oxaphospholenes by Neganova, Margarita E., Aleksandrova, Yulia R., Nikolaeva, Natalia S., Brel, Valery K.

“…[Display omitted] Using the methodology of “click” chemistry, a series of conjugates of 3,5-bis(benzylidene)-1-(prop-2-yn)piperidin-4-ones with…”
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Manganese(II) Thiocyanate Complexes with Bis(phosphine Oxide) Ligands: Synthesis and Excitation Wavelength‐Dependent Multicolor Luminescence by Davydova, Maria P., Bauer, Irina A., Brel, Valery K., Rakhmanova, Mariana I., Bagryanskaya, Irina Yu, Artem'ev, Alexander V.

“…First examples of luminescent MnII thiocyanate complexes are presented. A series of such compounds has been synthesized via the reaction of Mn(NCS)2 with…”
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Synthesis and antitumor activity of daunorubicin conjugates with of 3,4-methylendioxybenzaldehyde by Moiseeva, Aleksandra A., Artyushin, Oleg I., Anikina, Lada V., Brel, Valery K.

“…[Display omitted] The design of hybrid (chimeric) molecules containing two different pharmacophores connected via a spacer (linker) is a promising approach to…”
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New Approach toward Dual-Emissive Organic–Inorganic Hybrids by Integrating Mn(II) and Cu(I) Emission Centers in Ionic Crystals by Artem’ev, Alexander V., Davydova, Maria P., Berezin, Alexey S., Samsonenko, Denis G., Bagryanskaya, Irina Yu, Brel, Valery K., Hei, Xiuze, Brylev, Konstantin A., Artyushin, Oleg I., Zelenkov, Lev E., Shishkin, Ivan I., Li, Jing

“…Inorganic–organic hybrid luminescent materials have received great attention for their potential applications in a wide range of clean/renewable energy-related…”
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Low-symmetry A3B type pentachlorocyclotriphosphazene substituted phthalocyanine with improved nonlinear optical properties: Synthesis, spectroscopic and ab initio/(TD)DFT study by Tolbin, Alexander Yu, Brel, Valery K., Tarasevich, Boris N., Pushkarev, Victor E.

“…In the present work, we performed structural modification of 2-hydroxy-9(10),16(17),23(24)-tri-tert-butyl-29H,31H-phthalocyanine (1) using phosphonitrilic…”
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Synthesis and biological evaluation of indolylglyoxylamide bisphosphonates, antimitotic microtubule-targeting derivatives of indibulin with improved aqueous solubility by Brel, Valery K., Artyushin, Oleg I., Chuprov-Netochin, Roman N., Leonov, Sergey V., Semenova, Marina N., Semenov, Victor V.

“…[Display omitted] Indibulin (D-24851) derivatives with bisphosphonate fragment connected to the N1 atom of imidazole ring were synthesized by alkylation of…”
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Synthesis of camphecene derivatives using click chemistry methodology and study of their antiviral activity by Artyushin, Oleg I., Sharova, Elena V., Vinogradova, Natalya M., Genkina, Galina K., Moiseeva, Aleksandra A., Klemenkova, Zinaida S., Orshanskaya, Iana R., Shtro, Anna A., Kadyrova, Renata A., Zarubaev, Vladimir V., Yarovaya, Olga I., Salakhutdinov, Nariman F., Brel, Valery K.

“…[Display omitted] A series of seventeen tetrazole derivatives of 1,7,7-trimethyl-[2.2.1]bicycloheptane were synthesized using click chemistry methodology and…”
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Copper(I)‐Arsine Clusters with a Near‐Unity Phosphorescence Quantum Yield for X‐Ray Scintillation and LED Applications by Demyanov, Yan V., Ma, Zihao, Jia, Zhenglin, Rakhmanova, Marianna I., Carignan, Gia M., Bagryanskaya, Irina Yu, Sulyaeva, Veronika S., Globa, Anastasiya A., Brel, Valery K., Meng, Lingqiang, Meng, Hong, Lin, Qianqian, Li, Jing, Artemev, Alexander V.

“…Rare‐earth element‐free materials that exhibit strong room temperature phosphorescence (RTP) and X‐ray scintillation properties are gaining global interest…”
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Synthesis of Camphecene and Cytisine Conjugates Using Click Chemistry Methodology and Study of Their Antiviral Activity by Artyushin, Oleg. I., Moiseeva, Aleksandra A., Zarubaev, Vladimir V., Slita, Aleksander V., Galochkina, Anastasiya V., Muryleva, Anna A., Borisevich, Sophia S., Yarovaya, Olga I., Salakhutdinov, Nariman F., Brel, Valery K.

“…A series of camphecene and quinolizidine alkaloid (−)‐cytisine conjugates has been obtained for the first time using ‘click’ chemistry methodology. The…”
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Design, synthesis and antiviral evaluation of novel conjugates of the 1,7,7‐trimethylbicyclo[2.2.1]heptane scaffold and saturated N‐heterocycles via 1,2,3‐triazole linker by Sokolova, Anastasiya S., Yarovaya, Olga I., Artyushin, Oleg I., Sharova, Elena V., Baev, Dmitriy S., Mordvinova, Ekaterina D., Shcherbakov, Dmitriy N., Shnaider, Tatiana A., Nikitina, Tatiana V., Esaulkova, Iana L., Ilyina, Polina A., Zarubaev, Vladimir V., Brel, Valery K., Tolstikova, Tatyana G., Salakhutdinov, Nariman F.

“…A new series of heterocyclic derivatives with a 1,7,7‐trimethylbicyclo[2.2.1]heptane fragment was designed, synthesised and biologically evaluated. Synthesis…”
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N-Phosphorylation of daunorubicin—synthetic approaches and antiproliferative properties of the products by Moiseeva, Aleksandra A., Artyushin, Oleg I., Anikina, Lada V., Klemenkova, Zinaida S., Brel, Valery K.

“…Synthetic approaches to daunorubicin derivatives containing azide and propargyl fragments were developed. A series of phosphonate and bisphosphonate…”
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New tripodal ligand on the triphenylphosphine oxide platform with 1,2,3-triazole side arms: synthesis, structure, coordination, and extraction properties by Kudryavtsev, Igor Y., Bykhovskaya, Olga V., Matveeva, Anna G., Baulina, Tatyana V., Pasechnik, Margarita P., Matveev, Sergey V., Vologzhanina, Anna V., Turanov, Alexander N., Karandashev, Vasilii K., Brel, Valery K.

“…New hybrid tripodal propeller ligands on the triphenylphosphine oxide platform with triazole rings in the side arms and alkyl and aryl substituents in the…”
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Simple methods of modification of daunorubicin on the daunosamine nitrogen atom by Brel, Valery K., Moiseeva, Aleksandra A., Artyushin, Oleg I., Anikina, Lada V., Klemenkova, Zinaida S.

“…Modification of daunorubicin on its NH 2 moiety is a well-established synthetic approach to obtain novel derivatives of this compound. Moreover, the…”
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Synthesis of 2H-azirinyl phosphonates and phosphine oxides from phosphorus containing allenes by Brel, Valery K., Kovaleva, Ekaterina Yu, Nelyubina, Yulia V.

“…New 1,2-alkadienylphosphonates and diphenyl(1,2-alkadien-1-yl)phosphine oxides were synthesized by a convenient and efficient method. These compounds are…”
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Functionalization of bioactive substrates with a F5SCH = CH moiety by Brel, Valery K., Artyushin, Oleg I., Moiseeva, Aleksandra A., Sharova, Elena V., Buyanovskaya, Anastasiya G., Nelyubina, Yulia V.

“…A convenient approach to modify bioactive substrates such as daunorubicin, cytisine, and camphecene with a pentafluorosulfanylvinyl moiety have been suggested…”
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Synthesis, Structure, and Luminescence Properties of a {Mo6I8} Complex with (C6F5)2PO2 Ligands by Mironova, Alina D., Mikhajlov, Maxim A., Sukhikh, Taisiya S., Brylev, Konstantin A., Gushchin, Artem L., Eltsov, Ilia V., Stass, Dmitri V., Goryunov, Evgeny I., Brel, Valery K., Sokolov, Maxim N.

“…Reaction of [Mo6I8(CH3COO)6]2– with bis(pentafluorophenyl)phosphinic acid HO(O)P(C6F5)2 yielded a new bright‐red luminescent complex [{Mo6I8}(O2P(C6F5)2)6]2–,…”
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3,5-Bis(Arylidene)-4-Piperidones Modified by Bisphosphonate Groups as Novel Anticancer Agents by Makarov, Mikhail V., Rybalkina, Ekaterina Yu, Brel, Valery K.

“…Synthetic approaches for conjugating 3,5-bis(arylidene)-4-piperidones with bisphosphonate moiety were elaborated. These approaches are based either on reaction…”
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Synthesis of Alkene, Alcohols, and Heterocycles Containing the Pentafluorosulfanyl (SF5) Grouping by Brel, Valery K.

“…Convenient and effective methods for synthesis of heterocyclic derivatives with a pentafluorosulfanyl grouping have been presented…”
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New synthesis of trimethylsilyldiphenylphosphinite by Morgalyuk, Vasily P., Strelkova, Tat'yana V., Nifant'ev, Eduard E., Brel, Valery K.

“…A series of novel synthetically important reactions has been developed for the quick convenient and high-yield preparation of trimethylsilyl…”
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