Search Results - "Bourderioux, Aurelie"

Structural Basis for Inhibition of Mycobacterial and Human Adenosine Kinase by 7‑Substituted 7‑(Het)aryl-7-deazaadenine Ribonucleosides by Snášel, Jan, Nauš, Petr, Dostál, Jiří, Hnízda, Aleš, Fanfrlík, Jindřich, Brynda, Jiří, Bourderioux, Aurelie, Dušek, Michal, Dvořáková, Hana, Stolaříková, Jiřina, Zábranská, Helena, Pohl, Radek, Konečný, Petr, Džubák, Petr, Votruba, Ivan, Hajdúch, Marián, Řezáčová, Pavlína, Veverka, Václav, Hocek, Michal, Pichová, Iva

“…Adenosine kinase (ADK) from Mycobacterium tuberculosis (Mtb) was selected as a target for design of antimycobacterial nucleosides. Screening of…”
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Reactivity of tert-butanesulfinamides in palladium-catalyzed allylic substitutions by Mistico, Laetitia, Ay, Emel, Huynh, Vaizanne, Bourderioux, Aurelie, Chemla, Fabrice, Ferreira, Franck, Oble, Julie, Perez-Luna, Alejandro, Poli, Giovanni, Prestat, Guillaume

“…The performance of tert-butanesulfinamides as nitrogen nucleophiles in Pd(0)-catalyzed allylic substitution reactions has been investigated. Metalated N-alkyl…”
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Phosphine-Triggered Selectivity Switch in Silver-Catalyzed o‑Alkynylbenzohydroxamic Acid Cycloisomerizations by Bantreil, Xavier, Bourderioux, Aurélie, Mateo, Pierre, Hagerman, Caroline E, Selkti, Mohamed, Brachet, Etienne, Belmont, Philippe

“…A silver-catalyzed cycloisomerization reaction of a series of o-alkynylbenzohydroxamic acids is reported. Several 5-exo-dig and 6-endo-dig modes of cyclization…”
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Synthesis of new fused and substituted benzo and pyrido carbazoles via C-2 (het)arylindoles by Bourderioux, Aurélie, Kassis, Paméla, Mérour, Jean-Yves, Routier, Sylvain

“…In the course of a program aimed at designing new antitumor agents, we were interested in the synthesis of new substituted benzo and pyrido carbazoles. The…”
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Synthesis of benzo analogs of oxoarcyriaflavins and caulersine by Bourderioux, Aurélie, Routier, Sylvain, Bénéteau, Valérie, Mérour, Jean-Yves

“…In the course of a program aimed at designing new antitumor agents, we were interested in the synthesis of mixed structures of maleimidophenyl carbazoles and…”
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Synthesis and Significant Cytostatic Activity of 7-Hetaryl-7-deazaadenosines by Bourderioux, Aurelie, Nauš, Petr, Perlíková, Pavla, Pohl, Radek, Pichová, Iva, Votruba, Ivan, Džubák, Petr, Konečný, Petr, Hajdúch, Marián, Stray, Kirsten M, Wang, Ting, Ray, Adrian S, Feng, Joy Y, Birkus, Gabriel, Cihlar, Tomas, Hocek, Michal

“…A series of 7-aryl- and 7-hetaryl-7-deazaadenosines were prepared by the cross-coupling reactions of unprotected or protected 7-iodo-7-deazaadenosines with…”
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7-(2-Thienyl)-7-Deazaadenosine (AB61), a New Potent Nucleoside Cytostatic with a Complex Mode of Action by Perlíková, Pavla, Rylová, Gabriela, Nauš, Petr, Elbert, Tomáš, Tloušťová, Eva, Bourderioux, Aurelie, Slavětínská, Lenka Poštová, Motyka, Kamil, Doležal, Dalibor, Znojek, Pawel, Nová, Alice, Harvanová, Monika, Džubák, Petr, Šiller, Michal, Hlaváč, Jan, Hajdúch, Marián, Hocek, Michal

“…7-(2-Thienyl)-7-deazaadenosine (AB61) showed nanomolar cytotoxic activities against various cancer cell lines but only mild (micromolar) activities against…”
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Abstract 5100: AB61, a new potent nucleoside cytostatic: Molecular mechanisms of action and preclinical activity by Dzubak, Petr, Hajduch, Marian, Perlikova, Pavla, Rylová, Gabriela, Naus, Petr, Elbert, Tomas, Tloustova, Eva, Bourderioux, Aurelie, Slavetinska, Lenka, Motyka, Kamil, Dolezal, Dalibor, Znojek, Pawel, Nova, Alice, Harvanova, Monika, Siler, Michal, Hlavac, Jan, Hocek, Michal

“…Abstract 7-(2-Thienyl)-7-deazaadenosine (AB61) showed nanomolar cytotoxic activities against various cancer cell lines but only mild (micromolar) activities…”
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Sugar-modified derivatives of cytostatic 7-(het)aryl-7-deazaadenosines: 2′-C-methylribonucleosides, 2′-deoxy-2′-fluoroarabinonucleosides, arabinonucleosides and 2′-deoxyribonucleosides by Nauš, Petr, Perlíková, Pavla, Bourderioux, Aurelie, Pohl, Radek, Slavětínská, Lenka, Votruba, Ivan, Bahador, Gina, Birkuš, Gabriel, Cihlář, Tomáš, Hocek, Michal

“…A series of novel sugar-modified derivatives of cytostatic 7-hetaryl-7-deazaadenosines (2′-C-methylribonucleosides, 2′-deoxy-2′-fluoroarabinonucleosides,…”
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Synthesis and biological evaluation of novel oxophenylarcyriaflavins as potential anticancer agents by Bourderioux, Aurélie, Bénéteau, Valérie, Mérour, Jean-Yves, Baldeyrou, Brigitte, Ballot, Caroline, Lansiaux, Amélie, Bailly, Christian, Le Guével, Rémy, Guillouzo, Christiane, Routier, Sylvain

“…We report the synthesis and biological evaluation of new oxophenylarcyriaflavins designed as potential anticancer agents. An efficient synthesis involving…”
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Sugar-modified derivatives of cytostatic 7-(het)aryl-7-deazaadenosines: 2a2-C-methylribonucleosides, 2a2-deoxy-2a2-fluoroarabinonucleosides, arabinonucleosides and 2a2-deoxyribonucleosides by Naus, Petr, Perlikova, Pavla, Bourderioux, Aurelie, Pohl, Radek, Slavtinska, Lenka, Votruba, Ivan, Bahador, Gina, Birkus, Gabriel, Cihlac, Tomas, Hocek, Michal

“…A series of novel sugar-modified derivatives of cytostatic 7-hetaryl-7-deazaadenosines (2a2-C-methylribonucleosides, 2a2-deoxy-2a2-fluoroarabinonucleosides,…”
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Phosphine-Triggered Selectivity Switch in Silver-Catalyzed o -Alkynylbenzohydroxamic Acid Cycloisomerizations by Bantreil, Xavier, Bourderioux, Aurélie, Mateo, Pierre, Hagerman, Caroline, Selkti, Mohamed, Brachet, Etienne, Belmont, Philippe

“…A silver-catalyzed cycloisomerization reaction of a series of o-alkynylbenzohydroxamic acids is reported. Several 5-exo-dig and 6-endo-dig modes of cyclization…”
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Corrigendum to “Synthesis of new fused and substituted benzo and pyrido carbazoles via C-2 (het)arylindoles” [Tetrahedron 64(49) (2008) 11012–11019] by Bourderioux, Aurélie, Kassis, Paméla, Mérour, Jean-Yves, Routier, Sylvain

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The glucosinolate-myrosinase system. New insights into enzyme-substrate interactions by use of simplified inhibitors by Bourderioux, Aurélie, Lefoix, Myriam, Gueyrard, David, Tatibouét, Arnaud, Cottaz, Sylvain, Arzt, Steffi, Burmeister, Wim P, Rollin, Patrick

“…Myrosinase, a thioglucoside glucohydrolase, is the only enzyme able to hydrolyse glucosinolates, a unique family of molecules bearing an anomeric O-sulfated…”
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First efficient synthesis of novel oxophenyl-arcyriaflavin analogs by Bourderioux, Aurélie, Routier, Sylvain, Bénéteau, Valérie, Mérour, Jean-Yves

“…New oxophenylarcyriaflavins were synthesized in a few efficient steps. The key steps involved at first a palladium cross-coupling between the 3-bromo-4-(1…”
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