Search Results - "Bouillon, Marc"

Diastereoselective concise syntheses of the polyhydroxylated alkaloids DMDP and DAB by Bouillon, Marc E., Pyne, Stephen G.

“…A diastereoselective concise synthesis of the iminosugars DMDP and DAB is presented starting from l-xylose and affording the two alkaloids in good yields of…”
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The 4.4′-benzidine rearrangement of 4-alkyl substituted hydrazobenzenes by Bouillon, Marc E., Meyer, Hartmut H.

“…When treated with dilute inorganic acids N,N′-diarylhydrazines (hydrazobenzenes) with an alkyl substituent in the 4-position undergo [5,5]-sigmatropic…”
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Improving the antiprotozoal effect of saponins in the rumen by combination with glycosidase inhibiting iminosugars or by modification of their chemical structure by Ramos-Morales, Eva, de la Fuente, Gabriel, Nash, Robert J, Braganca, Radek, Duval, Stephane, Bouillon, Marc E, Lahmann, Martina, Newbold, C Jamie

“…The antiprotozoal effect of saponins is transitory, as when saponins are deglycosylated to sapogenins by rumen microorganisms they become inactive. We…”
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Synthesis of Anemoclemosides A and B, Two Saponins Isolated from Anemoclema glaucifolium by Bouillon, Marc E., Bertocco, Katia, Bischoff, Laura, Buri, Michelle, Davies, Lucy R., Wilkinson, Elizabeth J., Lahmann, Martina

“…Steroidal and triterpenoid saponins are attractive for their wide‐ranging pharmacological properties. The triterpenoid saponins Anemoclemoside A and B are root…”
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Modified Hederagenin Derivatives Demonstrate Ex Vivo Anthelmintic Activity against Fasciola hepatica by Chakroborty, Anand, Pritchard, Deiniol R, Bouillon, Marc E, Cervi, Anna, Kraehenbuehl, Rolf, Wild, Charlotte, Fenn, Caroline, Holdsworth, Peter, Capner, Colin, Padalino, Gilda, Forde-Thomas, Josephine E, Payne, Joseph, Smith, Brendan G, Fisher, Maggie, Lahmann, Martina, Baird, Mark S, Hoffmann, Karl F

“…Infection with (liver fluke) causes fasciolosis (or fascioliasis) and poses a considerable economic as well as welfare burden to both the agricultural and…”
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Flukicidal effects of abietane diterpenoid derived analogues against the food borne pathogen Fasciola hepatica by Chakroborty, Anand, Pritchard, Deiniol, Bouillon, Marc E., Cervi, Anna, Cookson, Alan, Wild, Charlotte, Fenn, Caroline, Payne, Joseph, Holdsworth, Peter, Capner, Colin, O’Neill, Jenna, Padalino, Gilda, Forde-Thomas, Josephine, Gupta, Sandeep, Smith, Brendan G., Fisher, Maggie, Lahmann, Martina, Baird, Mark S., Hoffmann, Karl F.

“…Control of liver fluke infections remains a significant challenge in the livestock sector due to widespread distribution of drug resistant parasite…”
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Concise synthesis of (-)-steviamine and analogues and their glycosidase inhibitory activities by Jiangseubchatveera, Nadechanok, Bouillon, Marc E, Liawruangrath, Boonsom, Liawruangrath, Saisunee, Nash, Robert J, Pyne, Stephen G

“…A concise synthesis of (-)-steviamine is reported along with the synthesis of its analogues 10-nor-steviamine, 10-nor-ent-steviamine and 5-epi-ent-steviamine…”
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An investigation of the antileishmanial properties of semi-synthetic saponins by Anderson, Orlagh, Beckett, Joseph, Briggs, Carla C, Natrass, Liam A, Cranston, Charles F, Wilkinson, Elizabeth J, Owen, Jack H, Mir Williams, Rhodri, Loukaidis, Angelos, Bouillon, Marc E, Pritchard, Deiniol, Lahmann, Martina, Baird, Mark S, Denny, Paul W

“…Leishmaniasis is a neglected tropical disease caused by insect-vector borne protozoan parasites of the, Leishmania species. Whilst infection threatens and…”
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Novel olanzapine analogues presenting a reduced H1 receptor affinity and retained 5HT2A/D2 binding affinity ratio by Jafari, Somayeh, Bouillon, Marc E, Huang, Xu-Feng, Pyne, Stephen G, Fernandez-Enright, Francesca

“…Olanzapine is an atypical antipsychotic drug with high clinical efficacy, but which can cause severe weight gain and metabolic disorders in treated patients…”
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Studies towards the synthesis of polyhydroxylated pyrrolidine alkaloids isolated from Broussonetia kazinoki (moraceae) by Bouillon, Marc E., Nash, Robert J., Pyne, Stephen G.

“…The syntheses of L-AB1, L-DMDP, and the novel compounds, (−)-phenethyl-L-AB1, (−)-10′-deoxobroussonetine C, (−)-10′-deoxobroussonetine E,…”
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Antiprotozoal Effect of Saponins in the Rumen Can Be Enhanced by Chemical Modifications in Their Structure by Ramos-Morales, Eva, de la Fuente, Gabriel, Duval, Stephane, Wehrli, Christof, Bouillon, Marc, Lahmann, Martina, Preskett, David, Braganca, Radek, Newbold, Charles J

“…The antiprotozoal effect of saponins is transitory, as when saponins are deglycosylated to the sapogenin by rumen microorganisms they become inactive. We…”
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Modified Hederagenin Derivatives Demonstrate Ex Vivo Anthelmintic Activity against IFasciola hepatica/I by Chakroborty, Anand, Pritchard, Deiniol R, Bouillon, Marc E, Cervi, Anna, Kraehenbuehl, Rolf, Wild, Charlotte, Fenn, Caroline, Holdsworth, Peter, Capner, Colin, Padalino, Gilda, Forde-Thomas, Josephine E, Payne, Joseph, Smith, Brendan G, Fisher, Maggie, Lahmann, Ma, Baird, Mark S, Hoffmann, Karl F

“…Infection with Fasciola hepatica (liver fluke) causes fasciolosis (or fascioliasis) and poses a considerable economic as well as welfare burden to both the…”
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Diastereoselective total synthesis of (+)-morusimic acid B, an amino acid from Morus alba by Bouillon, Marc E., Meyer, Hartmut H.

“…An efficient, flexible and diastereoselective synthesis of the naturally occurring pyrrolidine amino acid, (+)-morusimic acid B, has been accomplished…”
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An investigation of the antileishmanial properties of semi-synthetic saponins† †Electronic supplementary information (ESI) available. See DOI: 10.1039/d0md00123f by Anderson, Orlagh, Beckett, Joseph, Briggs, Carla C., Natrass, Liam A., Cranston, Charles F., Wilkinson, Elizabeth J., Owen, Jack H., Mir Williams, Rhodri, Loukaidis, Angelos, Bouillon, Marc E., Pritchard, Deiniol, Lahmann, Martina, Baird, Mark S., Denny, Paul W.

“…Hit anti-leishmanial saponin structures selected following primary and secondary screening. Leishmaniasis is a neglected tropical disease caused by…”
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Intent-Based Network Management with User-Friendly Interfaces and Natural Language Processing by Orlandi, Barbara, Lataste, Sandrine, Kerboeuf, Sylvaine, Bouillon, Marc, Huang, Xiaofeng, Faucheux, Frederic, Shahbazi, Arzhang, Delvallet, Pascal

“…This paper investigates the scaling of business ordering, delivery and fulfillment of 5G/6G services especially applied to network slicing. We propose a system…”
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A programmable and virtualized network & IT infrastructure for the internet of things: How can NFV & SDN help for facing the upcoming challenges by Omnes, Nathalie, Bouillon, Marc, Fromentoux, Gael, Le Grand, Olivier

“…The Internet of Things (IoT) revolution has major impacts on the network & Information Technology (IT) infrastructure. As IT in the past decade, network…”
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From a Business Intent to a Network Deployment with User-Friendly Interfaces and Natural Language Processing by Orlandi, Barbara, Lataste, Sandrine, Kerboeuf, Sylvaine, Bouillon, Marc, Huang, Xiaofeng, Marce, Olivier, Faucheux, Frederic, Cherrared, Sihem, Mongazon, Bruno, Delvallet, Pascal

“…Through a Proof-of-Concept, we illustrate how a business intent for ordering enterprise 5G services can be captured and fulfilled without need for telco…”
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Profit and Strategic Analysis for MNO-MVNO Partnership by Khalifa, Nesrine Ben, Benhamiche, Amal, Simonian, Alain, Bouillon, Marc

“…We consider a mobile market driven by two Mobile Network Operators (MNOs) and a new competitor Mobile Virtual Network Operator (MVNO). The MNOs can partner…”
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Profit and Strategic Analysis for MNO-MVNO Partnership by Khalifa, Nesrine Ben, Benhamiche, Amal, Simonian, Alain, Bouillon, Marc

“…We consider a mobile market driven by two Mobile Network Operators (MNOs) and a new competitor Mobile Virtual Network Operator (MVNO). The MNOs can partner…”
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