Search Results - "Bondarev, Mikhail L"

The medicinal chemistry of 5-HT6 receptor ligands with a focus on arylsulfonyltryptamine analogs by Glennon, Richard A, Siripurapu, Uma, Roth, Bryan L, Kolanos, Renata, Bondarev, Mikhail L, Sikazwe, Donald, Lee, Mase, Dukat, Małgorzata

“…Arylsulfonyl analogs of aminopyrimidines (e.g. Ro 04-6790; 2), aminopyridines (e.g. Ro 63-0563; 3), 1-phenylpiperazines (e.g. SB-271046; 4), and tryptamines…”
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Behavioral and biochemical investigations of bupropion metabolites by Bondarev, Mikhail L, Bondareva, Tatiana S, Young, Richard, Glennon, Richard A

“…The stimulus effects of bupropion metabolites were examined in a drug discrimination procedure using (−)nicotine- and (+)amphetamine-trained rats. (+)- and (−)…”
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Binding of amine-substituted N1-benzenesulfonylindoles at human 5-HT6 serotonin receptors by PULLAGURLA, Manik, SIRIPURAPU, Uma, KOLANOS, Renata, BONDAREV, Mikhail L, DUKAT, Małgorzata, SETOLA, V, ROTH, B. L, GLENNON, Richard A

“…An examination of several amine-substituted analogs of N(1)-benzenesulfonylindoles reveals that although they bind at human 5-HT(6) serotonin receptors with…”
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Preparation and Characterization of Lipophilic Doxorubicin Pro-drug Micelles by Li, Feng, Snow-Davis, Candace, Du, Chengan, Bondarev, Mikhail L, Saulsbury, Marilyn D, Heyliger, Simone O

“…Micelles have been successfully used for the delivery of anticancer drugs. Amphiphilic polymers form core-shell structured micelles in an aqueous environment…”
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Aminoalkoxyfluorenones and aminoalkoxybiphenyls: DNA binding modes by Zanoza, Svitlana O., Klimenko, Kyrylo O., Maltzev, George V., Bykova, Tetiana I., Levandovskiy, Igor A., Lyakhov, Sergiy A., Andronati, Sergiy A., Bondarev, Mikhail L.

“…[Display omitted] •Intercalation and minor groove binding are important for antiviral activity.•Planar fluorenones and nonplanar biphenyls were…”
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Binding of Sulfonyl-Containing Arylalkylamines at Human 5-HT6 Serotonin Receptors by Sikazwe, Donald, Bondarev, Mikhail L, Dukat, Małgorzata, Rangisetty, Jagadeesh B, Roth, Bryan L, Glennon, Richard A

“…Various sulfonyl-containing compounds (e.g. sulfonamides, sulfones) bind at human 5-HT6 serotonin receptors, but it has been difficult relating the binding…”
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β-Oxygenated Analogues of the 5-HT2A Serotonin Receptor Agonist 1-(4-Bromo-2,5-dimethoxyphenyl)-2-aminopropane by Glennon, Richard A, Bondarev, Mikhail L, Khorana, Nantaka, Young, Richard, May, Jesse A, Hellberg, Mark R, McLaughlin, Marsha A, Sharif, Najam A

“…Activation of 5-HT2A serotonin receptors represents a novel approach to lowering intraocular pressure. Because 5-HT2A serotonin receptor agonists might also…”
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PMMA-stimulus generalization to the optical isomers of MBDB and 3,4-DMA by Rangisetty, Jagadeesh B, Bondarev, Mikhail L, Chang-Fong, Jean, Young, Richard, Glennon, Richard A

“…Psychoactive phenylisopropylamines can produce one or more of several different stimulus effects in animals. These effects are typified by the hallucinogen…”
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Preparation and Characterization of Lipophilic Doxorubicin Pro-drug Micelles by Li, Feng, Snow-Davis, Candace, Du, Chengan, Bondarev, Mikhail L., Saulsbury, Marilyn D., Heyliger, Simone O.

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Binding of Sulfonyl-Containing Arylalkylamines at Human 5-HT 6 Serotonin Receptors by Sikazwe, Donald, Bondarev, Mikhail L., Dukat, Małgorzata, Rangisetty, Jagadeesh B., Roth, Bryan L., Glennon, Richard A.

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Binding of amine-substituted N 1-benzenesulfonylindoles at human 5-HT 6 serotonin receptors by Pullagurla, Manik, Siripurapu, Uma, Kolanos, Renata, Bondarev, Mikhail L., Dukat, Małgorzata, Setola, V., Roth, B.L., Glennon, Richard A.

“…Indoles 11 and 12 (R 1 and/or R 2 = NHCH 3 or H; R and R 3 = NH 2 or H) were examined to determine the influence of amine substituents on 5-HT 6 receptor…”
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β-Oxygenated Analogues of the 5-HT 2A Serotonin Receptor Agonist 1-(4-Bromo-2,5-dimethoxyphenyl)-2-aminopropane by Glennon, Richard A., Bondarev, Mikhail L., Khorana, Nantaka, Young, Richard, May, Jesse A., Hellberg, Mark R., McLaughlin, Marsha A., Sharif, Najam A.

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9-(Aminomethyl)-9,10-dihydroanthracene is a novel and unlikely 5-HT 2A receptor antagonist by Westkaemper, Richard B, Runyon, Scott P, Bondarev, Mikhail L, Savage, Jason E, Roth, Bryan L, Glennon, Richard A

“…Structural elaboration of phenylethylamine to 9-(aminomethyl)-9,10-dihydroanthracene (AMDA) produces an agent with high affinity ( K i=9.5–21 nM) at 5-HT 2A…”
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9-(Aminomethyl)-9,10-dihydroanthracene is a novel and unlikely 5-HT2A receptor antagonist by WESTKAEMPER, R. B, RUNYON, S. P, BONDAREV, M. L, SAVAGE, J. E, ROTH, B. L, GLENNON, R. A

“…Structural elaboration of phenylethylamine to 9-(aminomethyl)-9,10-dihydroanthracene (AMDA) produces an agent with high affinity (Ki = 9.5-21 nM) at 5-HT2A…”
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