Search Results - "Biradar, J S"

Synthesis, antioxidant and DNA cleavage activities of novel indole derivatives by Biradar, J.S., Sasidhar, B.S., Parveen, R.

“…A new series of novel indole derivatives containing barbitone moiety ( 5a- i) are synthesized by simple and efficient condensation of chalcones ( 3a- i) with…”
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Solvent-free, microwave assisted Knoevenagel condensation of novel 2,5-disubstituted indole analogues and their biological evaluation by Biradar, J.S., Sasidhar, B.S.

“…A rapid, efficient and environmental benign methodology for the preparation of 2,5-disubstituted indole analogues is developed. 2,5-Disubstituted…”
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Structural Elucidation of Alkaloids from Aerial Parts of Rivea hypocrateriformis and Their Antihemolytic and Cytotoxic Activity by Godipurge, S. S., Biradar, J. S., Biradar, N. J., Shivarudrappa, H. P., Yallappa, S., Hungund, B. S., Sreedhara Ranganath Pai, K.

“…Two new alkaloids, designated as hypocretine 1 and 2 , have been extracted from the aerial parts of Rivea hypocrateriformis, and their structures were…”
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A facile and green strategy for the synthesis of Au, Ag and Au–Ag alloy nanoparticles using aerial parts of R. hypocrateriformis extract and their biological evaluation by Godipurge, S.S., Yallappa, S., Biradar, Naveen J., Biradar, J.S., Dhananjaya, B.L., Hegde, Gajanan, Jagadish, K., Hegde, Gurumurthy

“…A facile and green strategy is reported here to synthesize gold (Au), silver (Ag) and gold–silver (Au–Ag) alloy nanoparticles (NPs) through bio-reduction…”
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Analysis of fluorescence quenching of new indole derivative by aniline using Stern–Volmer plots by Suresh Kumar, H.M., Kunabenchi, R.S., Biradar, J.S., Math, N.N., Kadadevarmath, J.S., Inamdar, S.R.

“…The fluorescence quenching of 5-methyl-3-phenyl-2-[4′-amino-s-triazolo-3′-yl] indole-5′-hydrazide (MPIH) by aniline quencher in cyclohexane, benzene, toluene…”
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Green Approach to the Synthesis of New Indole and Benzimidazole Analogs and Their Biological Evaluation by Rathod, A. S., Biradar, J. S.

“…To obtain new lead compounds with potent antimicrobial and antioxidant activities, new indole analogs containing various heterocyclic moieties were synthesized…”
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Synthesis of Some Indolyl Derivatives under Solvent Free Conditions, Their Cytotoxicity, and DNA Cleavage Studies by Rathod, A. S., Biradar, J. S.

“…A one-pot, rapid, facile, green, and efficient method of synthesis of pyran fused indolyl and 1,3-dicarbonyl analogs has been carried out under the…”
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An Efficient, Eco-Friendly Synthesis of Pyran Annulated Indole Analogs under Conventional Heating and Microwave Irradiation, and Their Anticancer and Antioxidant Activity by Rathod, A. S., Biradar, J. S.

“…A rapid, facile, green, eco-friendly, cost effective, and efficient method for the synthesis of pyran annulated indole analogs via one-pot, three components…”
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Microwave Assisted, Solvent-Free, “Green” Synthesis of Novel Indole Analogs as Potent Antitubercular and Antimicrobial Agents and Their Molecular Docking Studies by Rathod, A. S., Godipurge, S. S., Biradar, J. S.

“…A rapid, efficient and environmentally benign synthesis of novel indole analogs bearing thiazolidinone attached to substituted thiazolyl coumarin scaffolds are…”
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MK-10 Clay-Catalyzed Synthesis of 2-(2′,5′-Disubstituted-1′H-indol-3′-yl)-1H-benzo[d]imidazoles under Conventional and Microwave Irradiation by Biradar, J. S., Sharanbasappa, B.

“…The synthesis of benzimidazoles has been achieved in a one-pot reaction in excellent yield using a newly developed methodology. 2,5-Disubstituted-3-cyanoacetyl…”
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Potential transition state phosphoramidate inhibitors of β-tubulin as antifilarial agents by Anderson, R. J., Bendell, D. J., Hooper, M., Cairns, D., Mackay, S. P., Hiremath, S. P., Jivanagi, A. S., Badami, S., Biradar, J. S., Townson, S.

“…Transition state phosphoramidate inhibitors of β‐tubulin were designed as potential antifilarial agents. The reactionof 2‐aminobenzimidazole with diisopropyl…”
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Effect of Solvent Polarity on Fluorescence Quenching of New Indole Derivatives by CCl4 by Suresh Kumar, H. M., Kunabenchi, R. S., Nishti, S. V., Biradar, J. S., Kadadevarmath, J. S.

“…The fluorescence quenching of solutes 3-[5′-methyl-3′-phenylindol-2′-yl]-s-triazolo [3,4-b] [1,3,4] thiadiazol-6(5H)-thione (MPITTT) and…”
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Microwave-Assisted Synthesis of Some Indole and Isoniazid Derivatives as Antitubercular Agents and Molecular Docking Study by Rathod, A. S., Reddy, P. V., Biradar, J. S.

“…An efficient and expeditious microwave-assisted synthesis of isoniazid derivatives from various indole-3-carbaldehydes, phenols, and isoniazid via Betti’s…”
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Microwave-Assisted Synthesis of Some Indole and IsoniazidDerivatives as Antitubercular Agents and Molecular Docking Study by Rathod, A S, Reddy, P V, Biradar, J S

“…An efficient and expeditious microwave-assisted synthesis of isoniazid derivatives from various indole-3-carbaldehydes, phenols, and isoniazid via Betti’s…”
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SYNTHESIS, CHARACTERIZATION, AND BIOLOGICAL ACTIVITY OF NOVEL N-PHENYLPROPYL-3-SUBSTITUTED INDOLINE-2-ONE DERIVATIVES by ., Pushpa, Naraboli, Basavaraj S., Biradar, J. S.

“…Objective: The objective of the present work deals with the synthesis, characterization and evaluation of antimicrobial and antioxidant activity of…”
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Synthesis of some bisindolyl analogs for in vitro cytotoxic and DNA cleavage studies by Sasidhar, B. S., Biradar, J. S.

“…One-pot, three components, conventional and microwave-assisted synthesis of bisindolyl analogs is described. Michael addition of preformed 2,5-disubstituted…”
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DESIGN AND SYNTHESIS OF BENZODIAZEPINES BEARING BENZIMIDAZOLE/BENZOTHIAZOLE AND INDOLE MOIETIES AS A POTENT ANTIMICROBIAL AND ANTIOXIDANT AGENTS by Naraboli, Basavaraj Shivabasappa, Js, Biradar

“…  Objective: The present work deals with the synthesis and characterization of biologically active new indole derivatives, namely, 2-((1H-benzo[d]…”
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Synthesis and biological evaluation of novel Indolyl 4-thiazolidinones bearing thiadiazine nucleus by Anekal, Doddappa Pralhad, Biradar, J.S.

“…A series of Ethyl 2-[2-(2,5-disubstituted-1H-indol-3-yl)-4-oxothiazolid-3-ylamino]-5,6-dihydro-5-oxo-4H-1,3,4-thiadiazine-6-carboxylates (4a–g) were…”
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Effect of Solvent Polarity on Fluorescence Quenching of New Indole Derivatives by CCl 4 by Suresh Kumar, H. M., Kunabenchi, R. S., Nishti, S. V., Biradar, J. S., Kadadevarmath, J. S.

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