Search Results - "Bhondwe, Rahul S."

2‑(3-Fluoro-4-methylsulfonylaminophenyl)propanamides as Potent Transient Receptor Potential Vanilloid 1 (TRPV1) Antagonists: Structure–Activity Relationships of 2‑Amino Derivatives in the N‑(6-Trifluoromethylpyridin-3-ylmethyl) C‑Region by Kim, Myeong Seop, Ryu, HyungChul, Kang, Dong Wook, Cho, Seong-Hee, Seo, Sejin, Park, Young Soo, Kim, Mi-Yeon, Kwak, Eun Joo, Kim, Yong Soo, Bhondwe, Rahul S, Kim, Ho Shin, Park, Seul-gi, Son, Karam, Choi, Sun, DeAndrea-Lazarus, Ian A, Pearce, Larry V, Blumberg, Peter M, Frank, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Kögel, Babette Y, Schiene, Klaus, Christoph, Thomas, Lee, Jeewoo

“…A series of N-(2-amino-6-trifluoromethylpyridin-3-ylmethyl)-2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides were designed combining previously identified…”
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Structure–activity relationships and molecular modeling of the N-(3-pivaloyloxy-2-benzylpropyl)-N′-[4-(methylsulfonylamino)benzyl] thiourea template for TRPV1 antagonism by Bhondwe, Rahul S., Kang, Dong Wook, Kim, Myeong Seop, Kim, Ho Shin, Park, Seul-gi, Son, Karam, Choi, Sun, Lang Kuhs, Krystle A., Pavlyukovets, Vladimir A., Pearce, Larry V., Blumberg, Peter M., Lee, Jeewoo

“…The structure–activity relationships of N-(3-acyloxy-2-benzylpropyl)-N′-4-[(methylsulfonylamino)benzyl] thioureas, which represent simplified RTX-based…”
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N-4-t-Butylbenzyl 2-(4-methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure–activity relationships in the A-region by Kim, Yong Soo, Kil, Min-Jung, Kang, Sang-Uk, Ryu, HyungChul, Kim, Myeong Seop, Cho, Yongsung, Bhondwe, Rahul S., Thorat, Shivaji A., Sun, Wei, Liu, Keliang, Lee, Jin Hee, Choi, Sun, Pearce, Larry V., Pavlyukovets, Vladimir A., Morgan, Matthew A., Tran, Richard, Lazar, Jozsef, Blumberg, Peter M., Lee, Jeewoo

“…Structure–activity relationships for the A-region in a series of N-4-t-butylbenzyl 2-(4-methylsulfonylaminophenyl) propanamides as TRPV1 antagonists have been…”
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2-(4-Methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure–activity relationships in the B and C-regions by Sun, Wei, Liu, Keliang, Ryu, HyungChul, Kang, Dong Wook, Kim, Yong Soo, Kim, Myeong Seop, Cho, Yongsung, Bhondwe, Rahul S., Thorat, Shivaji A., Kim, Ho Shin, Pearce, Larry V., Pavlyukovets, Vladimir A., Tran, Richard, Morgan, Matthew A., Lazar, Jozsef, Ryder, Christopher B., Toth, Attila, Blumberg, Peter M., Lee, Jeewoo

“…On the basis of the previous lead N-4-t-butylbenzyl 2-(3-fluoro-4-methylsulfonylaminophenyl) propanamide (3) as a potent TRPV1 antagonist, structure–activity…”
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Structure-activity relationships and molecular modeling of the N-(3-pivaloyloxy-2-benzylpropyl)-Na2-[4-(methylsulfonylamino)benzy l] thiourea template for TRPV1 antagonism by Bhondwe, Rahul S, Kang, Dong Wook, Kim, Myeong Seop, Kim, Ho Shin, Park, Seul-gi, Son, Karam, Choi, Sun, Lang Kuhs, Krystle A, Pavlyukovets, Vladimir A, Pearce, Larry V, Blumberg, Peter M, Lee, Jeewoo

“…The structure-activity relationships of N-(3-acyloxy-2-benzylpropyl)-Na2-4-[(methylsulfonylamino)benzyl] thioureas, which represent simplified RTX-based…”
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