Search Results - "Bhalerao, Dinesh"

Synthesis of positional isomer and analogues of neostigmine methylsulfate: an anticholinesterase agent by Suresh, Chilamkurthi, Devi, Dharmasoth Rama, Basavaiah, Keloth, Prasada rao, K. V. V., Aegurla, Balakrishna, Kumar, Guduri Anil, Bhalerao, Dinesh, Kumar Reddy, Aaramadaka Sunil

“…The present research paper describes the origin, synthesis and characterization of a positional isomer and analogues of Neostigmine methylsulfate namely…”
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Synthesis and Process Optimization of Boceprevir: A Protease Inhibitor Drug by Bhalerao, Dinesh S, Arkala, Anil Kumar Reddy, Madhavi, Y. V, Nagaraju, M, Gade, Srinivas Reddy, Kumar, U. K. Syam, Bandichhor, Rakeshwar, Dahanukar, Vilas H

“…Efforts toward the synthesis and process optimization of boceprevir 1 are described. Boceprevir synthesis was optimized by telescoping the first three steps…”
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Oxidative Conversion of α,α-Disubstituted Acetamides to Corresponding One-Carbon-Shorter Ketones Using Hypervalent Iodine (λ5) Reagents in Combination with Tetraethylammonium Bromide by Bellale, Eknath V, Bhalerao, Dinesh S, Akamanchi, Krishnacharya G

“…α,α-Disubstituted acetamides undergo oxidative dehomologation to give one-carbon-shorter ketones when reacted with a hypervalent iodine (λ5) reagent in…”
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o-Iodoxybenzoic Acid- and Tetraethylammonium Bromide-Mediated Oxidative Transformation of Primary Carboxamides to One-Carbon Dehomologated Nitriles by Bhalerao, Dinesh S, Mahajan, Ulhas S, Chaudhari, Kiran H, Akamanchi, Krishnacharya G

“…A clean and efficient method for the oxidative transformations of primary carboxamides to one-carbon dehomologated nitriles using the combination of…”
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Mild and Efficient Method for [alpha]-Thiocyanation of Ketones and [beta]-Dicarbonyl Compounds Using Bromodimethylsulfonium Bromide-Ammonium Thiocyanate by Bhalerao, Dinesh S, Akamanchi, Krishnacharya G

“…An efficient and convenient method for α-thiocyanation of ketones and [beta]-dicarbonyl compounds has been developed using a reagent combination of…”
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First Total Synthesis of N-(3-Guanidinopropyl)-2-(4-hydroxyphenyl)-2-oxoacetamide by More, Satish S., Raghunadh, Akula, Shankar, Ramanathan, Patel, Navin B., Bhalerao, Dinesh S., Syam Kumar, Unniaran K.

“…The first total synthesis of the α‐oxo amide‐based natural product, N‐(3‐guanidinopropyl)‐2‐(4‐hydroxyphenyl)‐2‐oxoacetamide (3), isolated from aqueous…”
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IBX/TEAB-mediated oxidative dimerization of thioamides: synthesis of 3,5-disubstituted 1,2,4-thiadiazoles by Patil, Pravin C., Bhalerao, Dinesh S., Dangate, Prasad S., Akamanchi, Krishnacharya G.

“…Thioamides undergo oxidative dimerization on treatment with hypervalent iodine(V)-containing reagents, particularly o-iodoxybenzoic acid (IBX), in the presence…”
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Ethenolate Transfer Reactions: A Facile Synthesis of Vinyl Esters by Kaliyaperumal Appaye, Srinivasan, Pandurang Nikumbh, Satish, Reddy Govindapur, Rajeshwar, Banerjee, Shyamapada, Bhalerao, Dinesh S., Syam Kumar, Unniaran K.

“…A simple and efficient metal‐free ethenolate transfer reaction has been elaborated in moderate‐to‐high yields from vinyl acetate. This reaction was…”
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Direct oxidative conversion of aldehydes to nitriles using IBX in aqueous ammonia by Arote, Nitin D., Bhalerao, Dinesh S., Akamanchi, Krishnacharya G.

“…A mild, simple, chemoselective and high yielding procedure for the direct oxidative conversion of aldehydes to nitriles has been developed using IBX in aqueous…”
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Novel Approach to the Synthesis of Omeprazole: An Antipeptic Ulcer Agent by Bhalerao, Dinesh S., Kondaiah, Golla China Mala, Dwivedi, Namrata, Mylavarappu, Ravi Kumar, Reddy, Lekkala Amarnath, Roy, Arnab, Nagaraju, Gudimalla, Reddy, Padi Pratap, Bhattacharya, Apurba, Bandichhor, Rakeshwar

“…A novel approach for the synthesis of omeprazole, a potent antiulcer drug, is described. The synthetic procedure involved the formation of an ester of the…”
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Oxidation of amidoximes with IBX and IBX/ TEAB by Deshmukh, Swapnil S., Huddar, Sameerana N., Bhalerao, Dinesh S., Akamanchi, and Krishnacharya G.

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Mild and Efficient Method for α-Thiocyanation of Ketones and β-Dicarbonyl Compounds Using Bromodimethylsulfonium Bromide-Ammonium Thiocyanate by Bhalerao, Dinesh S., Akamanchi, Krishnacharya G.

“…An efficient and convenient method for α -thiocyanation of ketones and β -dicarbonyl compounds has been developed using a reagent combination of…”
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Diastereoselective synthesis of a core fragment of ritonavir and lopinavir by Roy, Arnab, Reddy, Lekkala Amarnath, Dwivedi, Namrata, Naram, Jyothirmayi, Swapna, Rodda, Malakondaiah, Golla China, Ravikumar, Mylavarpu, Bhalerao, Dinesh, Pratap, Taduri Bhanu, Reddy, Padi Pratap, Bhattacharya, Apurba, Bandichhor, Rakeshwar

“…A novel approach to the synthesis of Boc-core, a key starting material for ritonavir and lopinavir involving an unprecedented diastereoselective nitroaldol…”
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Oxidative Bromination of Aromatic Compounds Using O-Iodoxybenzoic Acid with Tetraethylammonium Bromide by Bhalerao, Dinesh S., Mahajan, Ulhas S., Akamanchi, Krishnacharya G.

“…A mild and selective procedure for the bromination of activated arenes using o-iodoxybenzoic acid and tetraethylammonium bromide is presented. The reactions…”
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Oxidative Conversion of a,a-Disubstituted Acetamides to Corresponding One-Carbon-Shorter Ketones Using Hypervalent Iodine (λ5) Reagents in Combination with Tetraethylammonium Bromide by BELLALE, Eknath V, BHALERAO, Dinesh S, AKAMANCHI, Krishnacharya G

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Synthesis and Process Optimization of Amtolmetin: An Antiinflammatory Agent by Reddy, Lekkala Amarnath, Chakraborty, Saurya, Swapna, Rodda, Bhalerao, Dinesh, Malakondaiah, Golla China, Ravikumar, Mylavarapu, Kumar, Abhijeet, Reddy, Gade Srinivas, Naram, Jyothirmayi, Dwivedi, Namrata, Roy, Arnab, Himabindu, Vurimidi, Babu, Bangaru, Bhattacharya, Apurba, Bandichhor, Rakeshwar

“…Efforts toward the synthesis and process optimization of amtolmetin guacil 1 are described. High-yielding electrophilic substitution followed by Wolf−Kishner…”
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Parallel XML parsing by Bhalerao, Rohit Dinesh

“…XML has become a standard in representing semi-structured, tree-oriented documents. With ever increasing application domains its impact on distributed…”
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