Search Results - "Bezerra, Flávio A.F.M."

Synthesis and antitubercular activity of heteroaromatic isonicotinoyl and 7-chloro-4-quinolinyl hydrazone derivatives by Ferreira, Marcelle de L, Gonçalves, Raoni S B, Cardoso, Laura N de F, Kaiser, Carlos R, Candea, Andre L P, Henriques, Maria das Graças M de O, Lourenço, Maria C S, Bezerra, Flavio A F M, de Souza, Marcus V N

“…Two series of N'-(E)-heteroaromatic-isonicotinohydrazide derivatives (3a-f and 4a-b) and 1-(7-chloroquinolin-4-yl)-2-[(heteroaromatic)methylene]hydrazone…”
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Mefloquine–oxazolidine derivatives, derived from mefloquine and arenecarbaldehydes: In vitro activity including against the multidrug-resistant tuberculosis strain T113 by Gonçalves, Raoni S.B., Kaiser, Carlos R., Lourenço, Maria C.S., Bezerra, Flavio A.F.M., de Souza, Marcus V.N., Wardell, James L., Wardell, Solange M.S.V., Henriques, Maria das Graças M.de O., Costa, Thadeu

“…Ten new mefloquine–oxazolidine derivatives, 4-[(1S,8aR)-3-(aryl)hexahydro[1,3]oxazolo[3,4-a]pyridin-1-yl]-2,8-bis(trifluoromethyl)quinoline (1:…”
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Synthesis and antitubercular activity of 7-chloro-4-quinolinylhydrazones derivatives by Candéa, André L.P., Ferreira, Marcelle de L., Pais, Karla C., Cardoso, Laura N.de F., Kaiser, Carlos R., Henriques, Maria das Graças M.de O., Lourenço, Maria C.S., Bezerra, Flávio A.F.M., de Souza, Marcus V.N.

“…A series of twenty-one quinoline derivatives have been synthesized and evaluated against Mycobacterium tuberculosis. Three compounds exhibited a significant…”
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Synthesis of α- and β-Pyran Naphthoquinones as a New Class of Antitubercular Agents by Ferreira, Sabrina B., de Carvalho da Silva, Fernando, Bezerra, Flávio A. F. M., Lourenço, Maria C. S., Kaiser, Carlos R., Pinto, Angelo C., Ferreira, Vitor F.

“…A series of α‐ and β‐pyran naphthoquinones (lapachones) have been synthesized and evaluated for their in‐vitro antibacterial activity against Mycobacterium…”
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Anti-Tuberculosis Evaluation and Conformational Study of N-Acylhydrazones Containing the Thiophene Nucleus by Cardoso, Laura N. F., Bispo, Marcelle L. F., Kaiser, Carlos R., Wardell, James L., Wardell, Solange M. S. V., Lourenço, Maria C. S., Bezerra, Flávio A. F. M., Soares, Rodrigo P. P., Rocha, Marcele N., de Souza, Marcus V. N.

“…A series of N‐acylhydrazonyl‐thienyl derivatives (compounds 2 and 3), mainly of the type 2‐(aryl‐CHNNHCOCH2)‐thiene (2: aryl = substituted‐phenyl; 3: aryl =…”
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Anti-Mycobacterial Evaluation of 7-Chloro-4-Aminoquinolines and Hologram Quantitative Structure-Activity Relationship (HQSAR) Modeling of Amino-Imino Tautomers by Bispo, Marcelle L F, Lima, Camilo H S, Cardoso, Laura N F, Candéa, André L P, Bezerra, Flávio A F M, Lourenço, Maria C S, Henriques, Maria G M O, Alencastro, Ricardo B, Kaiser, Carlos R, Souza, Marcus V N, Albuquerque, Magaly G

“…In an ongoing research program for the development of new anti-tuberculosis drugs, we synthesized three series ( , , and ) of 7-chloro-4-aminoquinolines, which…”
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