Search Results - "Berger, Michael L."

Lapses of the Heart: Frequency and Subjective Salience of Impressions Reported by Patients after Cardiac Arrest by Sterz, Fritz, Berger, Michael L, Ruzicka, Gerhard, Beisteiner, Roland

“…After cardiac arrest (CA), some patients report impressions with highly realistic features, often referred to as near-death experience (NDE). The frequency of…”
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Disturbed neurotransmitter homeostasis in ether lipid deficiency by Dorninger, Fabian, König, Theresa, Scholze, Petra, Berger, Michael L, Zeitler, Gerhard, Wiesinger, Christoph, Gundacker, Anna, Pollak, Daniela D, Huck, Sigismund, Just, Wilhelm W, Forss-Petter, Sonja, Pifl, Christian, Berger, Johannes

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NMDA receptor affinities of 1,2-diphenylethylamine and 1-(1,2-diphenylethyl)piperidine enantiomers and of related compounds by Berger, Michael L., Schweifer, Anna, Rebernik, Patrick, Hammerschmidt, Friedrich

“…Open-chain analogues of the prominent NMDA channel blocker MK-801 exhibit a high degree of stereoselectivity, inhibiting the binding of [ 3H]MK-801 to rat…”
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GABA(A) receptor subtype-selectivity of novel bicuculline derivatives by Ramerstorfer, Joachim, Foppa, Verena, Thiery, Hanna, Hermange, Philippe, Janody, Simon, Berger, Michael L, Dodd, Robert H, Sieghart, Werner

“…GABA(A) receptors are the major inhibitory neurotransmitter receptors in the central nervous system and are targets of clinically important drugs modulating…”
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Holographic Quantitative Structure-Activity Relationships of Tryptamine Derivatives at NMDA, 5HT1A and 5HT2A Receptors by Palangsuntikul, Rungtiva, Berner, Heinz, Berger, Michael, Wolschann, Peter

“…Tryptamine derivatives (Ts) were found to inhibit the binding of [3H]MK-801, [3H]ketanserin and [3H]8-OH-DPAT to rat brain membranes. [3H]MK-801 labels the…”
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Development and automation of a novel NET-PET tracer: [11 C]Me@APPI by Mark, Christina, Bornatowicz, Birgit, Mitterhauser, Markus, Hendl, Matthias, Nics, Lukas, Haeusler, Daniela, Lanzenberger, Rupert, Berger, Michael L, Spreitzer, Helmut, Wadsak, Wolfgang

“…Abstract Introduction The norepinephrine transporter (NET) is an important target for research in neurology and psychology and is involved in the…”
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Disturbed neurotransmitter homeostasis in ether lipid deficiency by Dorninger, Fabian, König, Theresa, Scholze, Petra, Berger, Michael L, Zeitler, Gerhard, Wiesinger, Christoph, Gundacker, Anna, Pollak, Daniela D, Huck, Sigismund, Just, Wilhelm W, Forss-Petter, Sonja, Pifl, Christian, Berger, Johannes

“…Plasmalogens, the most prominent ether (phospho)lipids in mammals, are structural components of most cellular membranes. Due to their physicochemical…”
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Soaping the NMDA receptor: Various types of detergents influence differently [3H]MK-801 binding to rat brain membranes by Berger, Michael L.

“…Membranes prepared from rat brain were treated with increasing concentrations of cationic, neutral, anionic and zwitterionic surfactants. Potent inactivation…”
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Synthesis of Thieno[2,3-b]Pyridinones Acting as Cytoprotectants and as Inhibitors of [3H]Glycine Binding to the N-Methyl-d-aspartate (NMDA) Receptor by Buchstaller, Hans-Peter, Siebert, Carsten D, Steinmetz, Ralf, Frank, Ina, Berger, Michael L, Gottschlich, Rudolf, Leibrock, Joachim, Krug, Michael, Steinhilber, Dieter, Noe, Christian R

“…The standard glycine site antagonist of the N-methyl-d-aspartate (NMDA) receptor, 3-phenyl-4-hydroxyquinolin-2(1H)-one (21), was used as a template for…”
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On the 'Stickiness' of Words. A Comparative Language Study Screening the Internet for English, German, French and Latin Phrases by Berger, Michael L.

“…Language, one of the defining attributes of Homo sapiens, not only deploys as a chain of words. Rather, words group together in a non-random way to form…”
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Differential influence of 7 cations on 16 non-competitive NMDA receptor blockers by Berger, Michael L., Rebernik, Patrick

“…[Display omitted] The specific binding of the NMDA receptor (NR) channel ligand [3H]MK-801 to rat brain membranes is sensitive to positively charged buffer…”
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New polyamine-sensitive inhibitors of the NMDA receptor: Syntheses and pharmacological evaluation by Pöhler, Thomas, Schadt, Oliver, Niepel, Daniela, Rebernik, Patrick, Berger, Michael L., Noe, Christian R.

“…Derivatives of 5-(4-aminobutyl)-2-thiophene-octylamine, a potent polyamine-sensitive inhibitor of the NMDA receptor, were synthesized and evaluated as…”
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Zinc regulates the dopamine transporter in a membrane potential and chloride dependent manner by Pifl, Christian, Wolf, Alexandra, Rebernik, Patrick, Reither, Harald, Berger, Michael L.

“…The dopamine transporter (DAT), a membrane protein specifically expressed by dopaminergic neurons and mediating the action of psychostimulants and dopaminergic…”
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Pentamidine analogs as inhibitors of [3H]MK-801 and [3H]ifenprodil binding to rat brain NMDA receptors by Berger, Michael L., Maciejewska, Dorota, Vanden Eynde, Jean Jacques, Mottamal, Madhusoodanan, Żabiński, Jerzy, Kaźmierczak, Paweł, Rezler, Mateusz, Jarak, Ivana, Piantanida, Ivo, Karminski-Zamola, Grace, Mayence, Annie, Rebernik, Patrick, Kumar, Arvind, Ismail, Mohamed A., Boykin, David W., Huang, Tien L.

“…[Display omitted] The anti-protozoal drug pentamidine is active against opportunistic Pneumocystis pneumonia, but in addition has several other biological…”
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Structure–activity relationship of etomidate derivatives at the GABAA receptor: Comparison with binding to 11β-hydroxylase by Atucha, Erika, Hammerschmidt, Friedrich, Zolle, Ilse, Sieghart, Werner, Berger, Michael L.

“…Two modifications of metomidate [(R)-1] without influence on inhibition of [131I]4-I-(R)-1 binding to 11β-hydroxylase reduced inhibitory potency at the GABAA…”
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Holographic quantitative structure-activity relationships of tryptamine derivatives at NMDA, 5HT(1A) and 5HT(2A) receptors by Palangsuntikul, Rungtiva, Berner, Heinz, Berger, Michael L, Wolschann, Peter

“…Tryptamine derivatives (Ts) were found to inhibit the binding of [³H]MK-801, [³H]ketanserin and [³H]8-OH-DPAT to rat brain membranes. [³H]MK-801 labels the…”
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New Selective Inhibitors of Steroid 11β-Hydroxylation in the Adrenal Cortex. Synthesis and Structure–Activity Relationship of Potent Etomidate Analogues by Zolle, Ilse M, Berger, Michael L, Hammerschmidt, Friedrich, Hahner, Stefanie, Schirbel, Andreas, Peric-Simov, Biljana

“…Derivatives of etomidate were evaluated as inhibitors of adrenal steroid 11β-hydroxylations. Stereoselective coupling by Mitsunobu produced chirally pure…”
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Exploring the Polyamine Regulatory Site of the NMDA Receptor: a Parallel Synthesis Approach by Berger, Michael L., Pöhler, Thomas, Schadt, Oliver, Stanger, Maximilian, Rebernik, Patrick, Scholze, Petra, Noe, Christian R.

“…The elongated structures of polyamine inverse agonists such as 1,12‐diaminododecane (N12N) and 5‐(4‐aminobutyl)‐2‐thiopheneoctanamine (N4T8N) lend themselves…”
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[3H]Metyrapol and 4‑[131I]Iodometomidate Label Overlapping, but Not Identical, Binding Sites on Rat Adrenal Membranes by Berger, Michael L, Hammerschmidt, Friedrich, Qian, Renzhe, Hahner, Stefanie, Schirbel, Andreas, Stichelberger, Martina, Schibli, Roger, Yu, Jie, Arion, Vladimir B, Woschek, Anna, Öhler, Elisabeth, Zolle, Ilse M

“…Metyrapone, metyrapol, and etomidate are competitive inhibitors of 11-deoxycorticosterone hydroxylation by 11β-hydroxylase. [3H]Metyrapol and…”
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New Selective Inhibitors of Steroid 11β-Hydroxylation in the Adrenal Cortex. Synthesis and Structure−Activity Relationship of Potent Etomidate Analogues by Zolle, Ilse M, Berger, Michael L, Hammerschmidt, Friedrich, Hahner, Stefanie, Schirbel, Andreas, Peric-Simov, Biljana

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