Search Results - "Bepary, Sukumar"
-
1
Synthesis of 2-Phenoxyacetic Acid Analogs for Evaluation of the Anti-inflammatory Potential and Subsequent In Silico Analysis
Published in Indonesian journal of chemistry (01-10-2024)“…Several 2-phenoxyacetic acid derivatives and their isosteres were synthesized in moderate to high yield (57–96%) for searching newer and safer alternatives to…”
Get full text
Journal Article -
2
Novel 3-amino-7-(aminomethyl)-1H-indazol-4-ol as the PI3Kγ enzyme inhibitor
Published in Bulletin of the Korean Chemical Society (01-12-2016)“…KCI Citation Count: 0…”
Get full text
Journal Article -
3
N-acetylation of 2-aminobenzothiazoles with Acetic Acid for Evaluation of Antifungal Activity and In Silico Analysis
Published in Journal of molecular docking (30-12-2021)“…Acetamides (S30A1 and S30) were synthesized from benzo[d]thiazol-2-amine and 6-nitrobenzo[d]thiazol-2-amine by direct use of acetic acid instead of acetylating…”
Get full text
Journal Article -
4
Rational design of novel diaryl ether-linked benzimidazole derivatives as potent and selective BACE1 inhibitors
Published in Biochemical and biophysical research communications (26-02-2024)“…Due to the large size and high flexibility of the catalytic active site of BACE1 enzyme, the development of nonpeptide inhibitors with optimal pharmacological…”
Get full text
Journal Article -
5
Novel 3‐amino‐7‐(aminomethyl)‐1 H ‐indazol‐4‐ol as the PI3Kγ enzyme inhibitor
Published in Bulletin of the Korean Chemical Society (01-12-2016)Get full text
Journal Article -
6
Synthesis of (3S,4S)-4-aminopyrrolidine-3-ol derivatives and biological evaluation for their BACE1 inhibitory activities
Published in Bioorganic & medicinal chemistry letters (01-01-2016)“…[Display omitted] Synthesis, SAR study and BACE1 inhibitory activity of (3S,4S)-4-aminopyrrolidine-3-ol derivatives (2) were described. The compound 7c…”
Get full text
Journal Article -
7
DPT-Mediated Synthesis of 2-Aminoimidazolidin-4-ones from Thioureas Tethered to Amides
Published in Synthetic communications (03-07-2014)“…2-Aminoimidazolidin-4-ones have been synthesized by using di-2-pyridyl thiocarbonate (DPT), taking the thioureas tethered to amides as the starting materials…”
Get full text
Journal Article -
8
Diversified Aminohydantoins from Ureas and Thioureas Tethered to Amides
Published in European journal of organic chemistry (01-05-2012)“…Intramolecular cyclization of thioureas or ureas tethered to amides afforded 2‐iminohydantoins and 2‐amino‐1H‐imidazol‐4(5H)‐ones in very high yields (87–100…”
Get full text
Journal Article -
9
Anti-inflammatory activity of indanyltetrazole derivatives
Published in Pakistan journal of pharmaceutical sciences (01-07-2008)“…A number of indanyl tetrazolederivatives namely 5-(6'-chloroindan-1'-yl)tetrazole (CIT), 5-(6'-bromoindan-1'-yl)tetrazole (BIT),…”
Get full text
Journal Article -
10
Report: in vitro dissolution studies of different brands of sustained release diclofenac sodium matrix tablet available in Bangladesh
Published in Pakistan journal of pharmaceutical sciences (01-01-2008)“…Commercially available national thirteen brands and three international brands of diclofenac sodium sustained release matrix tablets were studied in simulated…”
Get full text
Journal Article -
11
In vitro dissolution studies of different brands of sustained release diclofenac sodium matrix tablet available in Bangladesh
Published in Pakistan journal of pharmaceutical sciences (01-01-2008)“…Commercially available national thirteen brands and three international brands of diclofenac sodium sustained release matrix tablets were studied in simulated…”
Get full text
Journal Article -
12
Hepatoprotective activity of Phyllanthus reticulatus
Published in Pakistan journal of pharmaceutical sciences (01-10-2008)“…Two partially purified organic fractions designated by PR1 and PR2 of the fat free ethanol (95%) extract of aerial parts of Phyllanthus reticulatus were tested…”
Get full text
Journal Article