Search Results - "Bashiardes, G"

An expedient synthesis of diversified pyrrolizines and indolizines by Bashiardes, George, Safir, Imad, Barbot, Francis, Laduranty, Joelle

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A new method for the synthesis of plurisubstituted pyrroles by Bashiardes, George, Safir, Imad, Barbot, Francis, Laduranty, Joelle

“…A versatile method for the synthesis of pyrroles is described using an intramolecular [3+2] cycloaddition reaction. This method allows the expedient…”
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Microwave-Assisted [3 + 2] Cycloadditions of Azomethine Ylides by Bashiardes, George, Safir, Imad, Mohamed, Achmet Said, Barbot, Francis, Laduranty, Joelle

“…The microwave-assisted intramolecular [3 + 2] cycloaddition reaction of azomethine ylides to activated and nonactivated alkenes and alkynes is described. The…”
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Asymmetric Synthesis via Chiral Transition Metal Auxiliaries [and Discussion] by Davies, S. G., Bashiardes, G., Beckett, R. P., Coote, S. J., Dordor-Hedgecock, Isabelle M., Goodfellow, C. L., Gravatt, G. L., McNally, J. P., Whittaker, M., Reetz, M. T.

“…Stoichiometric reagents for the control of the absolute stereochemistry of new chiral centres produced during reactions involving carbon--carbon bond formation…”
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Synthesis and biological evaluation of a series of hydroxybenzylphenylamine derivatives as inhibitors of EGF receptor-associated tyrosine kinase activity by Chen, H, Bashiardes, G, Mailliet, P, Commercon, A, Sounigo, F, Boiziau, J, Parker, F, Tocque, B, Roques, B P, Garbay, C

“…In order to obtain non-degradable and more potent protein-tyrosine kinase inhibitors, derived from the 5-(2,5-dihydroxybenzyl)-aminosalicylates already…”
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Synthesis and phloem mobility of acidic derivatives of the fungicide fenpiclonil by Chollet, J.F, Rocher, F, Jousse, C, Deletage-Grandon, C, Bashiardes, G, Bonnemain, J.L

“…A series of derivatives of the phenylpyrrole fungicide fenpiclonil was synthesized in which a carboxyl group was present at various sites of this…”
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Acidic derivatives of the fungicide fenpiclonil: effect of adding a methyl group to the N-substituted chain on systemicity and fungicidal activity by Chollet, J.F, Rocher, F, Jousse, C, Deletage-Grandon, C, Bashiardes, G, Bonnemain, J.L

“…A new acidic derivative of the fungicide fenpiclonil was synthesized containing a methyl group on the alpha-position of the carboxyl function of…”
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Synthesis of non-immunosuppressive cyclophilin-binding cyclosporin A derivatives as potential anti-HIV-1 drugs by EVERS, Michel, BARRIERE, Jean-Claude, MIGNANI, Serge, BASHIARDES, Georges, BOUSSEAU, Anne, CARRY, Jean-Christophe, DEREU, Norbert, FILOCHE, Bruno, HENIN, Yvette, SABLE, Serge, VUILHORGNE, Marc

“…Original cyclosporin A (CsA) derivatives bearing various alkylthio side chains at the sarcosine residue 3 (R configuration) and for the most potent and…”
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Synthesis and biological evaluation of a new series of phenylhydroquinone derivatives as inhibitors of EGF-R-associated PTK activity by Million, M E, Mailliett, P, Chen, H, Bashiardes, G, Boiziau, J, Parker, F, Commerçon, A, Tocque, B, Roques, B P, Garbay, C

“…In order to design new potent inhibitors of the epidermal growth factor receptor (EGF-R) associated protein tyrosine kinase (PTK) activity as antitumor agents,…”
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The influence of organometallic chemistry on organic synthesis: present and future - Asymmetric synthesis via chiral transition metal auxiliaries by Davies, Stephen Graham, Bashiardes, G., Beckett, R. P., Coote, S. J., Dordor-Hedgecock, Isabelle M., Goodfellow, C. L., Gravatt, G. L., McNally, J. P., Whittaker, M.

“…Stoichiometric reagents for the control of the absolute stereochemistry of new chiral centres produced during reactions involving carbon-carbon bond formation…”
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