Search Results - "Barili, P"

Substituted 1,2,3-triazolo[1,5-a]quinazolines: synthesis and binding to benzodiazepine and adenosine receptors by Bertelli, Lucia, Biagi, Giuliana, Giorgi, Irene, Livi, Oreste, Manera, Clementina, Scartoni, Valerio, Lucacchini, Antonio, Giannaccini, Gino, Barili, Pier Luigi

“…This paper reports the synthesis and evaluation of the biological affinity towards benzodiazepine and A 1 and A 2A adenosine receptors of some 3-ethoxycarbonyl…”
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A Novel Class of Highly Potent and Selective A1 Adenosine Antagonists:  Structure−Affinity Profile of a Series of 1,8-Naphthyridine Derivatives by Ferrarini, Pier Luigi, Mori, Claudio, Manera, Clementina, Martinelli, Adriano, Mori, Filippo, Saccomanni, Giuseppe, Barili, Pier Luigi, Betti, Laura, Giannaccini, Gino, Trincavelli, Letizia, Lucacchini, Antonio

“…A series of 1,8-naphthyridine derivatives (12 − 36), bearing a phenyl group in position 2 and various substituents in positions 4 and 7, were synthesized in an…”
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1,2,3-Triazolo[1,5-a][1,4]- and 1,2,3-triazolo[1,5-a][1,5]benzodiazepine derivatives: synthesis and benzodiazepine receptor binding by Bertelli, Lucia, Biagi, Giuliana, Giorgi, Irene, Livi, Oreste, Manera, Clementina, Scartoni, Valerio, Martini, Claudia, Giannaccini, Gino, Trincavelli, Letizia, Barili, Pier Luigi

“…This paper reports the synthesis of new 1,2,3-triazolo[1,4]benzodiazepine and 1,2,3-triazolo[1,5]benzodiazepine derivatives and their evaluation toward…”
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1,2,3-Triazolo[1,5-a]quinoxalines: synthesis and binding to benzodiazepine and adenosine receptors by Bertelli, Lucia, Biagi, Giuliana, Giorgi, Irene, Manera, Clementina, Livi, Oreste, Scartoni, Valerio, Betti, Laura, Giannaccini, Gino, Trincavelli, Letizia, Barili, Pier Luigi

“…This paper reports the synthesis and binding assays toward benzodiazepine and adenosine A 1 and A 2A receptors of new 1,2,3-triazolo[1,5-a]quinoxalin-4-one…”
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Changes in the number of primary sensory neurons in normal and vitamin-E-deficient rats during aging by Cecchini, T, Cuppini, R, Ciaroni, S, Barili, P, De Matteis, R, Del Grande, P

“…In the dorsal root ganglia (DRGs) of vitamin-E-deficient rats, we previously found an increase in the number of neurons during the first 5 months of life…”
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Stereoselective synthesis and β-blocking activity of substituted (E)- and (Z)-4(1H)-[1-(3-alkylamino-2-hydroxypropyl)oximino]-2,3-dihydro-1,8-naphthyridine. Potential antihypertensive agents. Part VI by FERRARINI, P. L, MORI, C, BADAWNEH, M, MANERA, C, SACCOMANNI, G, CALDERONE, V, SCATIZZI, R, BARILI, P. L

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New 5-substituted-1-(2-hydroxybenzoyl)-benzotriazoles, potassium channel activators. IV by Biagi, Giuliana, Giorgi, Irene, Livi, Oreste, Scartoni, Valerio, Barili, Pier Luigi, Calderone, Vincenzo, Martinotti, Enrica

“…This paper reports the synthesis of a series of new 5-substituted-1-(2-hydroxybenzoyl)-benzotriazoles, which have been tested for their activity as possible…”
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4,6-O-benzylidene-D-glucopyranose and its sodium salt: new data on their preparation and properties by Barili, P L, Berti, G, Catelani, G, Cini, C, D'Andrea, F, Mastrorilli, E

“…An improved method for the preparation of 4,6-O-benzylidene-D-glucopyranose (BG), and new or correlated data on its 1H and 13C NMR spectra, specific rotations,…”
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Synthesis and benzodiazepine receptor activity of some 4,5-dihydro-1H-pyrazolo[4,3-c][1,8]naphthyridine derivatives by Da Settimo, A, Primofiore, G, Da Settimo, F, Simorini, F, Barili, P L, Senatore, G, Martini, C, Lucacchini, A

“…The preparation of 5-substituted 1-aryl-4,5-dihydro-1H-pyrazolo[4,3- c][1,8] naphthyridines by reaction of 5-substituted…”
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New syntheses of d-tagatose and of 1,5-anhydro- d-tagatose from d-galactose derivatives by Barili, Pier Luigi, Berti, Giancarlo, Catelani, Giorgio, D'Andrea, Felicia, Miarelli, Lucia

“…3,4- O-Isopropylidene- d- lyxo-hexopyranosid-2-ulose derivatives, obtained by oxidation of 3,4,6-protected d-galactopyranosides, can be alkylated in their…”
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1,2,3-triazole[4,5-d]pyridazines--IV. Preparation and adenosine receptor binding of new 4 and/or 7 aminoderivatives by Biagi, G, Giorgi, I, Livi, O, Scartoni, V, Velo, S, Martini, C, Senatore, G, Barili, P L

“…This paper reports the continuation of the studies on the 4-aminosubstituted 1,2,3-triazole[4,5-d]pyridazine derivatives which had shown binding affinity…”
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1,2,3-triazole[4,5-d]pyridazines. III--Synthesis of new 4-amino derivatives and their affinity toward adenosine receptors by Biagi, G, Giorgi, I, Livi, O, Scartoni, V, Lucacchini, A, Senatore, G, Barili, P L

“…This paper describes the preparation and adenosine receptor binding of new 1-benzyl-4-aminosubstituted-1,2,3-triazole[4,5-d]pyridazines and of other…”
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Structure-activity relationship studies in the field of calcium antagonists. Xanthone 1,4-dihydropyridines bearing a 2,3-lactone ring by Rampa, A, Budriesi, R, Bisi, A, Fabbri, G, Barili, P L, Chiarini, A, Valenti, P

“…A series of xanthone 1,4-dihydropyridine derivatives bearing a 2,3-lactone ring and a 2-acetoxymethyl group were prepared. The compounds were evaluated for…”
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Sensitivity to ageing of the limbic dopaminergic system: a review by Barili, Paolo, De Carolis, Gionni, Zaccheo, Damiano, Amenta, Francesco

“…The limbic system includes the complex of brain centres, nuclei and connections that provide the anatomical substrate for emotions. Although the presence of…”
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Dopamine D2-like receptors in the kidney of spontaneously hypertensive rats: a radioligand binding assay and light microscope autoradiography study by Barili, P, Fringuelli, C, Baldoni, E, Mignini, F, Zaccheo, D, Amenta, F

“…1. Dopamine D2-like receptors were investigated in sections of kidney from male spontaneously hypertensive rats (SHRs) at 6 and 14 weeks of age using…”
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A method for the synthesis of racemic and optically active 2-substituted 9-(2′,3′-dihydroxypropyl)-8-azahypoxanthines and 8-azaadenines by Barili, P. L., Biagi, G., Giorgi, I., Livi, O., Scartoni, V.

“…Several 9‐(2′,3′‐O‐isopropylidene)‐ and 9‐(2′,3′‐dihydroxypropyl)‐8‐azahypoxanthines and 8‐azaadenines were synthesized by a “one pot” method starting from the…”
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Microanatomical localization of dopamine receptor protein immunoreactivity in the rat cerebellar cortex by Barili, Paolo, Bronzetti, Elena, Ricci, Alberto, Zaccheo, Damiano, Amenta, Francesco

“…Dopamine (DA) receptor subtype localization was investigated in rat cerebellar cortex using immunohistochemical techniques with antibodies raised against D1–D5…”
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Alkaline and enzymatic hydrolysis of isobutyl 3,4-anhydro-2,6-dideoxy-DL-hexopyranosides. Preparation of enantiomeric boivinopyranosides through a highly efficient kinetic resolution by Barili, Pier Luigi, Berti, Giancarlo, Catelani, Giorgio, Colonna, Fabrizia, Mastrorilli, Ettore

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Structure-activity relations in cinnamamides. 1. Synthesis and pharmacological evaluation of some (E)- and (Z)-N-alkyl-.alpha.,.beta.-dimethylcinnamamides by Balsamo, A, Barili, P. L, Crotti, P, Macchia, B, Macchia, F, Pecchia, A, Cuttica, A, Passerini, N

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A facile "one pot" synthesis of 2,9-disubstituted 8-azapurin-6-ones (3,5-disubstituted 7-hydroxy-3H-1,2,3-triazolo[4,5-d]pyrimidines) by Barili, Pier Luigi, Biagi, Giuliana, Livi, Oreste, Scartoni, Valerio

“…A series of title compounds have been synthesized by utilising benzylazide, cyanoacetamide, ethyl or methyl esters of aliphatic or aromatic carboxylic acids…”
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