Search Results - "Bakulev, Vasiliy A."

Differentiation between Isomeric 4,5-Functionalized 1,2,3-Thiadiazoles and 1,2,3-Triazoles by ESI-HRMS and IR Ion Spectroscopy by Mazur, Dmitrii M, Piacentino, Elettra L, Berden, Giel, Oomens, Jos, Ryzhov, Victor, Bakulev, Vasiliy A, Lebedev, Albert T

“…A large variety of 1,2,3-thiadiazoles and 1,2,3-triazoles are used extensively in modern pure and applied organic chemistry as important structural blocks of…”
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Synthesis, Fungicidal Activity and Plant Protective Properties of 1,2,3-Thiadiazole and Isothiazole-Based N -acyl- N -arylalaninates by Kalinina, Tatiana A, Balandina, Valeriya I, Obydennov, Konstantin L, Slepukhin, Pavel A, Fan, Zhijin, Bakulev, Vasiliy A, Glukhareva, Tatiana V

“…The addition of active groups of known fungicides, or systemic acquired resistance inducers, into novel compound molecules to search for potential antifungal…”
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[3+2] Anionic Cycloaddition of Isocyanides to Acyclic Enamines and Enaminones: A New, Simple, and Convenient Method for the Synthesis of 2,4‐Disubstituted Pyrroles by Efimov, Ilya V., Matveeva, Maria D., Luque, Rafael, Bakulev, Vasiliy A., Voskressensky, Leonid G.

“…We herein demonstrate a new approach for the synthesis of 2,4‐disubstituted pyrroles by [3+2] cycloaddition reaction of isocyanides to the activated double…”
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Synthesis of Non-Aromatic Pyrroles Based on the Reaction of Carbonyl Derivatives of Acetylene with 3,3-Diaminoacrylonitriles by Silaichev, Pavel S, Dianova, Lidia N, Beryozkina, Tetyana V, Berseneva, Vera S, Maslivets, Andrey N, Bakulev, Vasiliy A

“…The reaction of 3,3-diaminoacrylonitriles with DMAD and 1,2-dibenzoylacetylene was studied. It is shown that the direction of the reaction depends on the…”
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Cyanothioacetamides as a synthetic platform for the synthesis of aminopyrazole derivatives by Filimonov, Valeriy O, Topchiy, Alexandra I, Ilkin, Vladimir G, Beryozkina, Tetyana V, Bakulev, Vasiliy A

“…It was shown that the reaction of 2-cyanothioacetamides with hydrazine involves both cyano- and thioamide groups, and 3,5-diaminopyrazoles are formed. In the…”
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Cycloaddition reactions of heterocyclic azides with 2-cyanoacetamidines as a new route to C , N -diheteroarylcarbamidines by Silaichev, Pavel S, Beryozkina, Tetyana V, Melekhin, Vsevolod V, Filimonov, Valeriy O, Maslivets, Andrey N, Ilkin, Vladimir G, Dehaen, Wim, Bakulev, Vasiliy A

“…A novel and efficient base-catalyzed, transition-metal-free method for the synthesis of diheterocyclic compounds connected by an amidine linker, including…”
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The Rich Chemistry Resulting from the 1,3‐Dipolar Cycloaddition Reactions of Enamines and Azides by Bakulev, Vasiliy A., Beryozkina, Tetyana, Thomas, Joice, Dehaen, Wim

“…Enamines exhibit exceptionally high reactivity in their 1,3‐dipolar cycloaddition reactions with azides in comparison with other dipolarophiles. This review…”
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Selective Synthesis of Azoloyl NH-1,2,3-Triazoles and Azolyl Diazoketones: Experimental and Computational Insights by Shafran, Yuri M, Hussein, Aqeel A, Beliaev, Nikolai A, Shevyrin, Vadim A, Shityakov, Sergey, Beryozkina, Tetyana V, Bakulev, Vasiliy A

“…Here, we report that the reaction of enaminones, from a class of azole series, with sulfonyl azides leads to a difficult-to-separate mixture of two pairs of…”
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Rh(II)-mediated domino [4 + 1]-annulation of α-cyanothioacetamides using diazoesters: A new entry for the synthesis of multisubstituted thiophenes by Medvedev, Jury J, Efimov, Ilya V, Shafran, Yuri M, Suslonov, Vitaliy V, Bakulev, Vasiliy A, Nikolaev, Valerij A

“…A new approach towards the synthesis of multisubstituted thiophenes is elaborated based on Rh(II)-catalyzed domino reactions of acyclic diazoesters with…”
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Design, Synthesis, and Evaluation of the Antifungal Activity of Novel Pyrazole–Thiazole Carboxamides as Succinate Dehydrogenase Inhibitors by Yu, Bin, Zhou, Shuang, Cao, Lixin, Hao, Zesheng, Yang, Dongyan, Guo, Xiaofeng, Zhang, Nailou, Bakulev, Vasiliy A, Fan, Zhijin

“…Succinate dehydrogenase (SDH) is regarded as a promising target for fungicide discovery. To continue our ongoing studies on the discovery of novel SDH…”
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Exploration of Fungicidal Activity and Mode of Action of Ferimzone Analogs by Zhang, Yue, Li, Jing, Liu, Xiaoyu, Gao, Wei, Song, Shuoshuo, Rong, Yaping, Tan, Linyu, Glukhareva, Tatiana V., Bakulev, Vasiliy A., Fan, Zhijin

“…Lead discovery and molecular target identification are important for developing novel pesticides. Scaffold hopping, an effective approach of modern medicinal…”
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Combined experimental and theoretical studies of regio- and stereoselectivity in reactions of β-isoxazolyl- and β-imidazolyl enamines with nitrile oxides by Efimov, Ilya V, Shafikov, Marsel Z, Beliaev, Nikolai A, Volkova, Natalia N, Beryozkina, Tetyana V, Dehaen, Wim, Fan, Zhijin, Grishko, Viktoria V, Lubec, Gert, Slepukhin, Pavel A, Bakulev, Vasiliy A

“…Reactions of β-azolyl enamines and nitrile oxides were studied by both experimental and theoretical methods. ( )-β-(4-Nitroimidazol-5-yl),…”
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Tandem Cycloaddition of Azides to 3,3-Diaminoacrylonitriles (2-Cyanoacetamidines) and Cornforth-Type Rearrangement as an Approach to 5‑Amino-1,2,3-triazole-4‑N‑substituted Imidamides by Silaichev, Pavel S., Beryozkina, Tetyana V., Ilkin, Vladimir, Novikov, Mikhail S., Dehaen, Wim, Bakulev, Vasiliy A.

“…An efficient base-catalyzed, metal-free method for the synthesis of 5-amino-1,2,3-triazole-4-N-sulfonyl- and arylimidamides, directed by the structure of the…”
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Synthesis, Fungicidal Activity, and Molecular Docking of 2‑Acylamino and 2‑Thioacylamino Derivatives of 1H‑benzo[d]imidazoles as Anti-Tubulin Agents by Obydennov, Konstantin L, Kalinina, Tatiana A, Galieva, Nadezhda A, Beryozkina, Tetyana V, Zhang, Yue, Fan, Zhijin, Glukhareva, Tatiana V, Bakulev, Vasiliy A

“…This work deals with the synthesis and evaluation of fungicidal activity of benzimidazole derivatives, which are structural analogues of commercial…”
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Rhodium-Catalyzed Transannulation of 4,5-Fused 1‑Sulfonyl-1,2,3-triazoles with Nitriles. The Selective Formation of 1‑Sulfonyl-4,5-fused Imidazoles versus Secondary C–H Bond Migration by Ilkin, Vladimir G., Beryozkina, Tetyana V., Willocx, Daan, Silaichev, Pavel S., Veettil, Santhini Pulikkal, Dehaen, Wim, Bakulev, Vasiliy A.

“…The reactivity of readily available 4,5-fused-1-sulfonyl-1,2,3-triazoles was examined in the Rh­(II)-catalyzed transannulation reaction with nitriles. We have…”
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Synthesis of 1,2,3-Thiadiazole and Thiazole-Based Strobilurins as Potent Fungicide Candidates by Chen, Lai, Zhu, Yu-Jie, Fan, Zhi-Jin, Guo, Xiao-Feng, Zhang, Zhi-Ming, Xu, Jing-Hua, Song, Ying-Qi, Yurievich, Morzherin Y, Belskaya, Nataliya P, Bakulev, Vasiliy A

“…Strobilurin fungicides play a crucial role in protecting plants against different pathogens and securing food supplies. A series of 1,2,3-thiadiazole and…”
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A Base‐Controlled Reaction of 2‐Cyanoacetamidines (3,3‐Diaminoacrylonitriles) with Sulfonyl Azides as a Route to Nonaromatic 4‐Methylene‐1,2,3‐triazole‐5‐imines by Silaichev, Pavel S., Beryozkina, Tetyana V., Novikov, Mikhail S., Dehaen, Wim, Bakulev, Vasiliy A.

“…Reactions of 2‐cyanoacetamidines with sulfonyl azides were shown to take place via two different pathways to form a mixture of 1‐substituted…”
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Synthesis and properties of hydrazones bearing amide, thioamide and amidine functions by Belskaya, Nataliya P., Dehaen, Wim, Bakulev, Vasiliy A.

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A facile access for the synthesis of 1-hetero(aryl)-1,2,3-triazoles linked to equol under mild conditions by Nibin Joy, Muthipeedika, Beliaev, Nikolai, Beryozkina, Tetyana V., Bakulev, Vasiliy A.

“…We herein report a convenient methodology for the synthesis of 1-hetero(aryl)-1,2,3-triazoles linked with equol by utilizing copper-catalyzed azide-alkyne…”
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Thioisomünchnones versus Acrylamides via Copper-Catalyzed Reaction of Thioamides with Diazocarbonyl Compounds by Ilkin, Vladimir G., Filimonov, Valeriy O., Seliverstova, Eugenia A., Novikov, Mikhail S., Beryozkina, Tetyana V., Gagarin, Aleksey A., Belskaya, Nataliya P., Muthipeedika, Nibin Joy, Bakulev, Vasiliy A., Dehaen, Wim

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