Search Results - "Bakhmedova, A A"

Synthesis and cytotoxic properties of anomeric 5-substituted 3'-azido-2',3'-dideoxyuridines by Bakhmedova, A A, Iartseva, I V, Zhukova, O S, Volosiuk, T P, Iurkevich, A M, Mel'nik, S Ia

“…Glycosylation of trimethylsilyl derivatives of 5-benzyloxymethyl- and 5-hydroxymethyluracil with 3-azido-2,3-dideoxy-5-O-benzoyl-D-ribofuranosyl chloride…”
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The synthesis and and study of cytotoxic activity of D-ribofuranosides and 2-deoxy-D-ribofuranosides of substituted bis(indolyl)furan, -pyrrole and indolo[2,3-alphacarbazole derivatives by Garaeva, L D, Bakhmedova, A A, Iartseva, I V, Mel'nik, S Ia, Adanin, V M

“…1-(2,3,5-Tri-O-acetyl)-beta-D-ribofuranosyl indole, the key compound in the synthesis of glycosides with the bis(indole) aglycone, was obtained for the first…”
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Synthesis of potential antimetabolites in a series of carbohydrate-modified pyrimidine 2'-deoxynucleosides by Bakhmedova, A A, Iartseva, I V, Mel'nik, S Ia

“…The interaction of 3'-amino-2',3'-dideoxy- or 5'-amino-2',5'-dideoxy-5-substituted pyrimidine nucleosides with N-ethylmaleimide in DMF in the presence of Et3N…”
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Synthesis and antiproliferative properties of glycosides of bis(indolyl)furan-2,5-dione and bis(indolyl)-1H-pyrrol-2,5-dione by Mel'nik, S Ia, Bakhmedova, A A, Garaeva, L D, Goriunova, O V, Miniker, T D, Plikhtiak, I L, Ektova, L V, Iartseva, I V

“…A synthesis of the derivatives of bis(indolyl)furan and bis(indolyl)pyrrole, which contain an acyclic fragment or a residue of D-ribo-, D-xylo-, L-arabino-,…”
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Modulation of the antitumor activity of 1-(4-amino-2-methyl-5-pyrimidinyl)methyl-3-(2-chloroethyl)-3-nitrosoure a by O(6)-methyl-2'-deoxyguanosine--a new inhibitor of O(6)-alkylguanine-DNA-alkyltransferase by Dederer, L Iu, Sokolova, I S, Bakhmedova, A A, Miniker, T D, Mel'nik, S Ia, Gorbacheva, L B

“…O6-Methyl-2'-deoxyguanosine (O6-MedG), a novel inhibitor of O6-alkylguanine-DNA alkyltransferase (O6-AGT), has been synthesized. The ability of O6-MedG to…”
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Synthesis, conversion and biological activity of 5-substituted 2'-deoxyuridines modified by carbohydrates by Mel'nik, S Ia, Bakhmedova, A A, Iartseva, I V, Zhukova, O S, Iavorskaia, N P

“…5-Benzyloxymethyl(Bom)-2'-deoxyuridine and its alpha-anomer were used as the key compounds for syntheses of thymidine analogues or 3'-derivatives. Anomeric…”
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Synthesis and antiviral properties of anomeric 5-isopropoxymethyl and 5-(3-hydroxypropoxynethyl)-2′-desoxyurudines by Bakhmedova, A. A., Kochetkova, M. V., Yartseva, I. V., Chekunova, é. V., Mel'nik, S. Ya

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Search for antimetabolites among 5-trimethylsilyluracil nucleosides and their nonglycoside analogs by Mel'nik, S Ia, Bakhmedova, A A, Iartseva, I V, Preobrazhenskaia, M N, Zaguliaeva, O A, Mamaev, V P

“…The reaction of 2'-deoxy-5-trimethylsilyl(Tms)uridine with methanesulfonyl chloride led to the corresponding 3',5'-di-O-mesyl derivative, which was treated…”
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Synthesis and antimetabolite properties of 5-substituted 2'-deoxyuridines. Anomeric 5-(2-aminohexafluoroprop-2-yl)- and 5-(2-trifluoroacetylaminohexafluoroprop-2-yl)-2'-deoxyuridine by Mel'nik, S Ia, Bakhmedova, A A, Iartseva, I V, Kochetkova, M V, Preobrazhenskaia, M N

“…Alkylation of 2,4-bis-O-(trimethylsilyl)uracil with hexafluoroacetone trifluoroacetylimine gave 5-(2-trifluoroacelylaminohexafluoroprop-2-yl)uracil, which was…”
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Synthesis of anomeric 5-trimethylgermyl-2'-deoxyuridines and study of their antiviral and cytotoxic properties by Mel'nik, S Ia, Bakhmedova, A A, Nedorezova, T P, Iartseva, I V, Zhukova, O S

“…Glycosylation of silylated 5-trimethylgermyluracil with 2-deoxy-3,5-di-O-p-toluyl-alpha-D-ribofuranosylchloride in dichloroethane in the presence of SnCl4 and…”
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Synthesis and study of 5-(trialkylsilyl)pyrimidine nucleosides. A new alpha-2'-deoxynucleoside with antiherpes activity by Mel'nik, S Ia, Bakhmedova, A A, Miniker, T D, Iartseva, I V, Preobrazhenskaia, M N

“…Glycosylation of 5-trimethylsilyl- and 5-triethylsilyluracil as well as 5-trimethylsilylcytosine with 2-deoxy-3,5-di-O-p-toluyl-alpha-D-ribofuranosylchloride…”
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3-(1H-indol-3-yl)-4-(1-glykozylindol-3-yl)-1H-pyrrole-2,5-diones: synthesis and study of antiproliferative properties by Mel'nik, S Ia, Bakhmedova, A A, Garaeva, L D, Miniker, T D, Plikhtiak, I L, Ektova, L V, Ivanova, T P, Adanin, V M, Iartseva, I V

“…A synthesis of 3-(1H-3-indolyl)-4-(1-glycosyl-3-indolyl)furan-2,5-diones and -1H-pyrrole-2,5-diones modified with the residues of D-ribo-, D-xylo-, L-arabino-,…”
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Antiviral activity of anomeric 5-substituted 2'-deoxyuridines by Bektemirov, T A, Chekunova, E V, Andzhaparidze, O G, Mel'nik, S Ia, Bakhmedova, A A

“…The inhibiting effect for herpes and vaccinia viruses of 2'-deoxyuridine derivatives containing the substitute in the position of 5-pyrimidine ring was…”
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Phenanthrothiazoles: III. Synthesis of some phenanthro[3,4-d]thiazoles and determination of the structures of phenanthrothiazoles by means of PMR spectra by Bronovitskaya, V. P., Bakhmedova, A. A., Berlin, A. Ya, Alekseeva, L. M., Sheinker, Yu. N.

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