Search Results - "Baishya, Gakul"

A naturally derived small molecule disrupts ligand-dependent and ligand-independent androgen receptor signaling in human prostate cancer cells by Amin, Karishma S, Jagadeesh, Shankar, Baishya, Gakul, Rao, Paruchuri G, Barua, Nabin C, Bhattacharya, Samir, Banerjee, Partha P

“…Continued reliance on androgen receptor (AR) signaling is a hallmark of prostate cancer, including the development of castration-resistant prostate cancer…”
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Vapor of volatile oils from Litsea cubeba seed induces apoptosis and causes cell cycle arrest in lung cancer cells by Seal, Soma, Chatterjee, Priyajit, Bhattacharya, Sushmita, Pal, Durba, Dasgupta, Suman, Kundu, Rakesh, Mukherjee, Sandip, Bhattacharya, Shelley, Bhuyan, Mantu, Bhattacharyya, Pranab R, Baishya, Gakul, Barua, Nabin C, Baruah, Pranab K, Rao, Paruchuri G, Bhattacharya, Samir

“…Non-small cell lung carcinoma (NSCLC) is a major killer in cancer related human death. Its therapeutic intervention requires superior efficient molecule(s) as…”
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First Example of a Four‐Component Prins Cyclization Reaction: Diastereoselective Synthesis of Dithiocarbamate Derived Octahydro‐2H‐chromenes by Sarmah, Barnali, Baishya, Gakul, Das, Pranab J.

“…A novel one‐pot sequential four‐component Prins cyclization reaction has been developed for the synthesis of dithiocarbamate derived octahydro‐2H‐chromenes…”
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Hydrothiolation of Unactivated Alkynes Catalyzed by Indium(III) Bromide by Yadav, J. S, Reddy, B. V. Subba, Raju, A, Ravindar, K, Baishya, Gakul

“…Indium(III) bromide is found to catalyze efficiently the hydrothiolation of unactivated alkynes with various thiols under mild conditions to produce the…”
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Recent Advances in Direct C−H Trifluoromethylation of N‐Heterocycles by Baishya, Gakul, Dutta, Nibedita B.

“…Fluorine chemistry executes a vital role in the agricultural, pharmaceutical, and materials industries. Moreover, introducing fluorine atom and…”
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One-Pot Sequential Schmidt and Ritter Reactions for the Synthesis of N-tert-Butyl Amides by Hazarika, Nabajyoti, Baishya, Gakul

“…The first example of the direct conversion of benzaldehydes into their corresponding N‐tert‐butyl amides through a Schmidt reaction/Ritter reaction sequence is…”
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K2S2O8 mediated C-3 arylation of quinoxalin-2(1H)-ones under metal-, photocatalyst- and light-free conditions by Nibedita Baruah Dutta, Bhuyan, Mayurakhi, Baishya, Gakul

“…Two facile and effective C-3 arylation protocols of quinoxalin-2(1H)-ones with arylhydrazines and aryl boronic acids respectively via free radical…”
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Copper(II) Triflate Immobilized in [bmim]BF4 Ionic liquid: An Efficient Reaction Medium for Michael Addition of β-Ketoesters to Acceptor-activated Alkenes by Yadav, J. S, Reddy, B. V. S, Baishya, Gakul, Narsaiah, A. Venkat

“…1,3-Dicarbonyl compounds undergo smooth conjugate addition to α,β-unsaturated ketones in the presence of 10 mol % copper(II) triflate immobilized in air and…”
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K 2 S 2 O 8 mediated C-3 arylation of quinoxalin-2(1 H )-ones under metal-, photocatalyst- and light-free conditions by Dutta, Nibedita Baruah, Bhuyan, Mayurakhi, Baishya, Gakul

“…Two facile and effective C-3 arylation protocols of quinoxalin-2(1 )-ones with arylhydrazines and aryl boronic acids respectively free radical cross-coupling…”
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1-(Chloromethyl)-4-fluoro-1,4-diazoniabicyclo-[2,2,2]octane Bis(tetrafluoroborate) as Novel and Efficient Reagent for the Conjugate Addition of Indoles to α,β-Unsaturated Ketones by Yadav, J. S, Reddy, B. V. Subba, Raju, A, Ravindar, K, Baishya, Gakul

“…Indoles undergo smooth conjugate addition with α,β-unsaturated ketones in the presence of 10 mol % SelectfluorTM under extremely mild conditions to afford the…”
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K2S2O8 Mediated Three‐component Radical Cascade C3 Alkylation of Quinoxalin‐2(1H)‐ones with Vinylarenes and 4‐Hydroxycoumarins/4‐Hydroxy‐6‐methyl‐2‐pyrone by Sharma, Suraj, Bhuyan, Mayurakhi, Baishya, Gakul

“…Quinoxalin‐2(1H)‐ones undergo a three‐component radical cascade C3 alkylation reaction with 4‐hydroxycoumarins/4‐hydroxy‐6‐methyl‐2‐pyrone by using vinyl…”
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K 2 S 2 O 8 Mediated Three‐component Radical Cascade C3 Alkylation of Quinoxalin‐2(1 H )‐ones with Vinylarenes and 4‐Hydroxycoumarins/4‐Hydroxy‐6‐methyl‐2‐pyrone by Sharma, Suraj, Bhuyan, Mayurakhi, Baishya, Gakul

“…Quinoxalin‐2(1 H )‐ones undergo a three‐component radical cascade C3 alkylation reaction with 4‐hydroxycoumarins/4‐hydroxy‐6‐methyl‐2‐pyrone by using vinyl…”
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Pretreatment of hydroethanolic extract of Dillenia indica L. attenuates oleic acid induced NAFLD in HepG2 cells via modulating SIRT-1/p-LKB-1/AMPK, HMGCR & PPAR-α signaling pathways by Poornima, M.S., Sindhu, G., Billu, Abraham, Sruthi, C.R., Nisha, P., Gogoi, Pinku, Baishya, Gakul, G Raghu, K.

“…Dillenia indica L. is an edible plant from the Dilleniaceae family present in the forest of India and other Asian countries. Different parts of this plant are…”
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Metal‐, Photocatalyst‐, Light‐ and Electrochemical‐Free C‐3 Trifluoromethylation of Quinoxalin‐2(1H)‐ones, Imidazo[1,2‐a]pyridines and 2H‐Indazoles by Dutta, Nibedita Baruah, Bori, Jugal, Gogoi, Pinku, Baishya, Gakul

“…We report an efficient protocol for the synthesis of 3‐trifluoromethylquinoxalin‐2(1H)‐ones, 3‐trifluoromethylimidazo[1,2‐a]pyridines and…”
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Tyrosinase Inhibitory Kinetics, LC-QTOF-MS Based Chemical Profiling and Molecular Docking of Phytochemicals from Dillenia indica L. Barks by Gogoi, Pinku, Kumar, Amit, Das, Aparoop, Baishya, Gakul

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Prins–Arylthiolation Reaction on Terpenoids: Diastereoselective Synthesis of 4‐Arylthiooctahydro‐2 H ‐chromenes by Sarmah, Barnali, Baishya, Gakul, Baruah, Rajani K.

“…(–)‐Isopulegol undergoes Prins‐arylthiolation with different aldehydes and cyclohexanone in the presence of HBF 4 · OEt 2 to generate a library of…”
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KSO mediated C-3 arylation of quinoxalin-2(1)-ones under metal-, photocatalyst- and light-free conditions by Dutta, Nibedita Baruah, Bhuyan, Mayurakhi, Baishya, Gakul

“…Two facile and effective C-3 arylation protocols of quinoxalin-2(1 H )-ones with arylhydrazines and aryl boronic acids respectively via free radical…”
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HBF4·OEt2: An efficient fluorinated acid catalyst for the one-pot synthesis of secondary and tertiary N-homoallylic carbamates by Baishya, Gakul, Hazarika, Nabajyoti, Sarmah, Barnali

“…•HBF4·OEt2 is used as a catalyst for the first time in this reaction.•HBF4·OEt2 is used as superior alternative to metal triflates and other catalysts.•The…”
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Prins-Arylthiolation Reaction on Terpenoids: Diastereoselective Synthesis of 4-Arylthiooctahydro-2H-chromenes by Sarmah, Barnali, Baishya, Gakul, Baruah, Rajani K.

“…(–)‐Isopulegol undergoes Prins‐arylthiolation with different aldehydes and cyclohexanone in the presence of HBF4·OEt2 to generate a library of…”
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A Green Protocol for the Synthesis of α‐Diazo‐β‐hydroxyesters and One‐Pot Conversion to β‐Keto‐Esters and Imidazo[1,2‐a]pyridine‐3‐carboxylates by Dutta, Nibedita Baruah, Sharma, Suraj, Chetry, Rudra Lal, Baishya, Gakul

“…A new solvent cum reagent system comprising of water extract of banana ash and dimethylsulfoxide (WEB‐DMSO) has been engaged for the first time to promote the…”
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