Search Results - "BRADBURY, Annette E"

Non-covalent thrombin inhibitors featuring P3-Heterocycles with P1-Monocyclic arginine surrogates by REINER, John E, SIEV, Daniel V, GIBSON, Tony S, ANDERSON, Susanne M, BRADBURY, Annette E, NOLAN, Thomas G, SEMPLE, J. Edward, ARALDI, Gian-Luca, CUI, Jingrong Jean, HO, Jonathan Z, KOMANDLA MALLA REDDY, MAMEDOVA, Lala, VU, Phong H, LEE, Kuen-Shan S, MINAMI, Nathaniel K

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Non-covalent thrombin inhibitors featuring P3-heterocycles with P1-bicyclic arginine surrogates by CUI, Jingrong Jean, ARALDI, Gian-Luca, MINAMI, Nathaniel K, ANDERSON, Susanne M, BRADBURY, Annette E, NOLAN, Thomas G, SEMPLE, J. Edward, REINER, John E, KOMANDLA MALLA REDDY, KEMP, Scott J, HO, Jonathan Z, SIEV, Daniel V, MAMEDOVA, Lala, GIBSON, Tony S, GAUDETTE, John A

“…Novel, potent, and highly selective classes of thrombin inhibitors were identified, which resulted from judicious combination of P4-aromatics and…”
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Synthesis and biological activity of peptidyl aldehyde urokinase inhibitors by Tamura, S Y, Weinhouse, M I, Roberts, C A, Goldman, E A, Masukawa, K, Anderson, S M, Cohen, C R, Bradbury, A E, Bernardino, V T, Dixon, S A, Ma, M G, Nolan, T G, Brunck, T K

“…Solid- and solution-phase synthesis of peptidomimetic inhibitors of urokinase-type plasminogen activator based on the sequence dSerAlaArg-al are described. The…”
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Non-covalent thrombin inhibitors featuring p 3 -heterocycles with P 1 -monocyclic arginine surrogates by Reiner, John E, Siev, Daniel V, Araldi, Gian-Luca, Cui, Jingrong Jean, Ho, Jonathan Z, Reddy, Komandla Malla, Mamedova, Lala, Vu, Phong H, Lee, Kuen-Shan S, Minami, Nathaniel K, Gibson, Tony S, Anderson, Susanne M, Bradbury, Annette E, Nolan, Thomas G, Semple, J.Edward

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Non-covalent thrombin inhibitors featuring P(3)-heterocycles with P(1)-monocyclic arginine surrogates by Reiner, John E, Siev, Daniel V, Araldi, Gian Luca, Cui, Jingrong Jean, Ho, Jonathan Z, Reddy, Komandla Malla, Mamedova, Lala, Vu, Phong H, Lee, Kuen Shan S, Minami, Nathaniel K, Gibson, Tony S, Anderson, Susanne M, Bradbury, Annette E, Nolan, Thomas G, Semple, J Edward

“…Investigations on P(2)-P(3)-heterocyclic dipeptide surrogates directed towards identification of an orally bioavailable thrombin inhibitor led us to pursue…”
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