Search Results - "BIRKEMO, L. S"

The effects of anorectic and aversive agents on deprivation-induced feeding and taste aversion conditioning in rats by Ervin, G N, Birkemo, L S, Johnson, M F, Conger, L K, Mosher, J T, Menius, Jr, J A

“…We compared the effects of intraperitoneally administered LiCl (0.5-2830 mumol/kg), sulfated cholecystokinin26-33 (10-1000 nmol/kg; CCK-8), nonsulfated CCK-8…”
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Optimization of 3-(1H-Indazol-3-ylmethyl)-1,5-benzodiazepines as Potent, Orally Active CCK-A Agonists by Henke, Brad R, Aquino, Christopher J, Birkemo, Larry S, Croom, Dallas K, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, Hirst, Gavin C, James, Michael K, Johnson, Michael F, Queen, Kennedy L, Sherrill, Ronald G, Sugg, Elizabeth E, Suh, Edward M, Szewczyk, Jerzy W, Unwalla, Rayomand J, Yingling, Jeff, Willson, Timothy M

“…We previously described a series of 3-(1H-indazol-3-ylmethyl)-1,5-benzodiazepine CCK-A agonists exemplified by compound 1 (GW 5823), which is the first…”
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Modification of Receptor Selectivity and Functional Activity in Cholecystokinin Peptoid Ligands by Dezube, Milana, Sugg, Elizabeth E, Birkemo, Larry S, Croom, Dallas K, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, James, Michael K, Johnson, Michael F

“…Hybrid analogs of the cholecystokinin A (CCK-A) receptor selective tetrapeptide agonist Boc-Trp-Lys(Tac)-Asp-MePhe-NH2 (1,A-71623) and the CCK-B receptor…”
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3-(1H-indazol-3-ylmethyl)-1,5-benzo-diazepines : CCK-A agonists that demonstrate oral activity as satiety agents by HENKE, B. R, WILLSON, T. M, JAMES, M. K, SUGG, E. E, CROOM, D. K, DOUGHERTY, R. W, QUEEN, K. L, BIRKEMO, L. S, ERVIN, G. N, GRIZZLE, M. K, JOHNSON, M. T

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Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A) Receptor Agonist Activity. 1. Optimization of the Agonist “Trigger” by Aquino, Christopher J, Armour, Duncan R, Berman, Judd M, Birkemo, Larry S, Carr, Robin A. E, Croom, Dallas K, Dezube, Milana, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, Head, Julie E, Hirst, Gavin C, James, Michael K, Johnson, Michael F, Miller, Laurence J, Queen, Kennedy L, Rimele, Thomas J, Smith, David N, Sugg, Elizabeth E

“…Directed screening of compounds selected from the Glaxo registry file for contractile activity on the isolated guinea pig gallbladder (GPGB) identified a…”
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Sulfated Cholecystokinin [26–33]Induces Mild Taste Aversion Conditioning in Rats when Administered by Three Different Routes by Mosher, Jack T., Birkemo, Larry S., Johnson, Michael F., Ervin, Gregory N.

“…We investigated the ability of sulfated cholecystokinin [26–33](CCK-8) and cholecystokinin [30–33](CCK-4) to induce taste aversion or avoidance conditioning…”
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3-(1H-Indazol-3-ylmethyl)-1,5-benzodiazepines:  CCK-A Agonists That Demonstrate Oral Activity as Satiety Agents by Henke, Brad R, Willson, Timothy M, Sugg, Elizabeth E, Croom, Dallas K, Dougherty, Robert W, Queen, Kennedy L, Birkemo, Larry S, Ervin, Gregory N, Grizzle, Mary K, Johnson, Michael F, James, Michael K

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Multiple, small doses of cholecystokinin octapeptide are more efficacious at inducing taste aversion conditioning than single, large doses by Ervin, Gregory N., Mosher, Jack T., Birkemo, Larry S., Johnson, Michael F.

“…Using a one-bottle taste aversion conditioning paradigm, sulfated cholecystokinin(26–33) (CCK-8) has again been shown to induce taste aversion conditioning in…”
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Neurotensin blocks certain amphetamine-induced behaviours by Ervin, Gregory N, Birkemo, Larry S, Nemeroff, Charles B, Prange, Arthur J

“…Bilateral injections of either neurotensin (NT; 0.3, 1 or 5 micrograms in 1 microliter artificial CSF) or haloperidol (HA; 2.5 or 5 micrograms in 1 microliter…”
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Several roles of CCK sub(A) and CCK sub(B) receptor subtypes in CCK-8-induced and LiCl-induced taste aversion conditioning by Mosher, J T, Johnson, M F, Birkemo, L S, Ervin, G N

“…Administration of a relatively large IP dose of sulfated cholecystokinin (26-33) (CCK-8; 1.0 mu mol/kg) consistently induced moderate taste aversion…”
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Several roles of CCKA and CCKB receptor subtypes in CCK-8-induced and LiCl-induced taste aversion conditioning by Mosher, J T, Johnson, M F, Birkemo, L S, Ervin, G N

“…Administration of a relatively large IP dose of sulfated cholecystokinin (26-33) (CCK-8; 1.0 mumol/kg) consistently induced moderate taste aversion…”
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