Search Results - "BARILI, P. L"

Substituted 1,2,3-triazolo[1,5-a]quinazolines: synthesis and binding to benzodiazepine and adenosine receptors by Bertelli, Lucia, Biagi, Giuliana, Giorgi, Irene, Livi, Oreste, Manera, Clementina, Scartoni, Valerio, Lucacchini, Antonio, Giannaccini, Gino, Barili, Pier Luigi

“…This paper reports the synthesis and evaluation of the biological affinity towards benzodiazepine and A 1 and A 2A adenosine receptors of some 3-ethoxycarbonyl…”
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A Novel Class of Highly Potent and Selective A1 Adenosine Antagonists:  Structure−Affinity Profile of a Series of 1,8-Naphthyridine Derivatives by Ferrarini, Pier Luigi, Mori, Claudio, Manera, Clementina, Martinelli, Adriano, Mori, Filippo, Saccomanni, Giuseppe, Barili, Pier Luigi, Betti, Laura, Giannaccini, Gino, Trincavelli, Letizia, Lucacchini, Antonio

“…A series of 1,8-naphthyridine derivatives (12 − 36), bearing a phenyl group in position 2 and various substituents in positions 4 and 7, were synthesized in an…”
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1,2,3-Triazolo[1,5-a][1,4]- and 1,2,3-triazolo[1,5-a][1,5]benzodiazepine derivatives: synthesis and benzodiazepine receptor binding by Bertelli, Lucia, Biagi, Giuliana, Giorgi, Irene, Livi, Oreste, Manera, Clementina, Scartoni, Valerio, Martini, Claudia, Giannaccini, Gino, Trincavelli, Letizia, Barili, Pier Luigi

“…This paper reports the synthesis of new 1,2,3-triazolo[1,4]benzodiazepine and 1,2,3-triazolo[1,5]benzodiazepine derivatives and their evaluation toward…”
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Synthesis and benzodiazepine receptor activity of some 4,5-dihydro-1H-pyrazolo[4,3-c][1,8]naphthyridine derivatives by Da Settimo, A, Primofiore, G, Da Settimo, F, Simorini, F, Barili, P L, Senatore, G, Martini, C, Lucacchini, A

“…The preparation of 5-substituted 1-aryl-4,5-dihydro-1H-pyrazolo[4,3- c][1,8] naphthyridines by reaction of 5-substituted…”
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1,2,3-Triazolo[1,5-a]quinoxalines: synthesis and binding to benzodiazepine and adenosine receptors by Bertelli, Lucia, Biagi, Giuliana, Giorgi, Irene, Manera, Clementina, Livi, Oreste, Scartoni, Valerio, Betti, Laura, Giannaccini, Gino, Trincavelli, Letizia, Barili, Pier Luigi

“…This paper reports the synthesis and binding assays toward benzodiazepine and adenosine A 1 and A 2A receptors of new 1,2,3-triazolo[1,5-a]quinoxalin-4-one…”
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Structure-activity relationship studies in the field of calcium antagonists. Xanthone 1,4-dihydropyridines bearing a 2,3-lactone ring by Rampa, A, Budriesi, R, Bisi, A, Fabbri, G, Barili, P L, Chiarini, A, Valenti, P

“…A series of xanthone 1,4-dihydropyridine derivatives bearing a 2,3-lactone ring and a 2-acetoxymethyl group were prepared. The compounds were evaluated for…”
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Stereoselective synthesis and β-blocking activity of substituted (E)- and (Z)-4(1H)-[1-(3-alkylamino-2-hydroxypropyl)oximino]-2,3-dihydro-1,8-naphthyridine. Potential antihypertensive agents. Part VI by FERRARINI, P. L, MORI, C, BADAWNEH, M, MANERA, C, SACCOMANNI, G, CALDERONE, V, SCATIZZI, R, BARILI, P. L

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Structure-activity relations in cinnamamides. 1. Synthesis and pharmacological evaluation of some (E)- and (Z)-N-alkyl-.alpha.,.beta.-dimethylcinnamamides by Balsamo, A, Barili, P. L, Crotti, P, Macchia, B, Macchia, F, Pecchia, A, Cuttica, A, Passerini, N

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New 5-substituted-1-(2-hydroxybenzoyl)-benzotriazoles, potassium channel activators. IV by Biagi, Giuliana, Giorgi, Irene, Livi, Oreste, Scartoni, Valerio, Barili, Pier Luigi, Calderone, Vincenzo, Martinotti, Enrica

“…This paper reports the synthesis of a series of new 5-substituted-1-(2-hydroxybenzoyl)-benzotriazoles, which have been tested for their activity as possible…”
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4,6-O-benzylidene-D-glucopyranose and its sodium salt: new data on their preparation and properties by Barili, P L, Berti, G, Catelani, G, Cini, C, D'Andrea, F, Mastrorilli, E

“…An improved method for the preparation of 4,6-O-benzylidene-D-glucopyranose (BG), and new or correlated data on its 1H and 13C NMR spectra, specific rotations,…”
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New syntheses of d-tagatose and of 1,5-anhydro- d-tagatose from d-galactose derivatives by Barili, Pier Luigi, Berti, Giancarlo, Catelani, Giorgio, D'Andrea, Felicia, Miarelli, Lucia

“…3,4- O-Isopropylidene- d- lyxo-hexopyranosid-2-ulose derivatives, obtained by oxidation of 3,4,6-protected d-galactopyranosides, can be alkylated in their…”
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1,2,3-triazole[4,5-d]pyridazines--IV. Preparation and adenosine receptor binding of new 4 and/or 7 aminoderivatives by Biagi, G, Giorgi, I, Livi, O, Scartoni, V, Velo, S, Martini, C, Senatore, G, Barili, P L

“…This paper reports the continuation of the studies on the 4-aminosubstituted 1,2,3-triazole[4,5-d]pyridazine derivatives which had shown binding affinity…”
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1,2,3-triazole[4,5-d]pyridazines. III--Synthesis of new 4-amino derivatives and their affinity toward adenosine receptors by Biagi, G, Giorgi, I, Livi, O, Scartoni, V, Lucacchini, A, Senatore, G, Barili, P L

“…This paper describes the preparation and adenosine receptor binding of new 1-benzyl-4-aminosubstituted-1,2,3-triazole[4,5-d]pyridazines and of other…”
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A method for the synthesis of racemic and optically active 2-substituted 9-(2′,3′-dihydroxypropyl)-8-azahypoxanthines and 8-azaadenines by Barili, P. L., Biagi, G., Giorgi, I., Livi, O., Scartoni, V.

“…Several 9‐(2′,3′‐O‐isopropylidene)‐ and 9‐(2′,3′‐dihydroxypropyl)‐8‐azahypoxanthines and 8‐azaadenines were synthesized by a “one pot” method starting from the…”
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Alkaline and enzymatic hydrolysis of isobutyl 3,4-anhydro-2,6-dideoxy-DL-hexopyranosides. Preparation of enantiomeric boivinopyranosides through a highly efficient kinetic resolution by Barili, Pier Luigi, Berti, Giancarlo, Catelani, Giorgio, Colonna, Fabrizia, Mastrorilli, Ettore

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A facile "one pot" synthesis of 2,9-disubstituted 8-azapurin-6-ones (3,5-disubstituted 7-hydroxy-3H-1,2,3-triazolo[4,5-d]pyrimidines) by Barili, Pier Luigi, Biagi, Giuliana, Livi, Oreste, Scartoni, Valerio

“…A series of title compounds have been synthesized by utilising benzylazide, cyanoacetamide, ethyl or methyl esters of aliphatic or aromatic carboxylic acids…”
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"One pot" synthesis of 2,9-disubstituted 8-azaadenines (3,5-disubstituted 7-amino-3H-1,2,3-triazolo[4,5-d]pyrimidines) by Barili, Pier Luigi, Biagi, Giuliana, Livi, Oreste, Mucci, Luciana, Scartoni, Valerio

“…A new simple method for the synthesis of title compounds is described starting from malononitrile, benzyl‐azide and an aliphatic or aromatic nitrile…”
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Indane-1,3-dione, phthalimidine and phthalide derivatives as alkylating agents by Barili, Pier Luigi, Scartoni, Valerio

“…The title compounds gave carbocations in acid media. The electrophilic aromatic substitution of those carbocations was studied…”
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Nitrogen-15 magnetic resonance studies. Further evidence for the dependence of 1J(15NH) on the hybridization of nitrogen by Axenrod, Theodore, Wieder, M. J, Berti, Giancarlo, Barili, P. L

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Structure-activity relationship in cinnamamides. 2. Synthesis and pharmacological evaluation of some (E)- and (Z)-N-alkyl-alpha, beta-dimethylcinnamamides substituted on the phenyl group by Balsamo, A, Barili, P L, Crotti, P, Macchia, B, Macchia, F, Cuttica, A, Passerini, N

“…Several (E)- and (Z)-N-alkyl-alpha,beta-dimethylcinnamamides variously substituted on the phenyl group were synthesized from their corresponding acids and…”
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