Search Results - "BALDINO, C. M"

d,l- and meso-Isochrysohermidin : total synthesis and interstrand DNA cross-linking by BOGER, D. L, BALDINO, C. M

“…A concise total synthesis of isochrysohermidin (5) is detailed based on a novel application of the sym-tetrazine arrow right 1,2-diazine arrow right pyrrole…”
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Perspective Articles on the Utility and Application of Solution-Phase Combinatorial Chemistry by Baldino, Carmen M

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Microwave-assisted one-pot synthesis of 2,3-disubstituted 3H-quinazolin-4-ones by Liu, Ji-Feng, Lee, Jaekyoo, Dalton, Audra M., Bi, Grace, Yu, Libing, Baldino, Carmen M., McElory, Eric, Brown, Matt

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Regioselective synthesis of [1,2,3]-triazoles catalyzed by Cu(I) generated in situ from Cu(0) nanosize activated powder and amine hydrochloride salts by Orgueira, Hernán A., Fokas, Demosthenes, Isome, Yuko, Chan, Philip C.-M., Baldino, Carmen M.

“…[Display omitted] A straightforward and efficient method for the regioselective synthesis of functionalized 1,4-disubstituted [1,2,3]-triazoles, from terminal…”
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Novel One-Pot Total Syntheses of Deoxyvasicinone, Mackinazolinone, Isaindigotone, and Their Derivatives Promoted by Microwave Irradiation by Liu, Ji-Feng, Ye, Ping, Sprague, Kevin, Sargent, Katie, Yohannes, Daniel, Baldino, Carmen M, Wilson, Christopher J, Ng, Shi-Chung

“…Total syntheses of deoxyvasicinone (1), mackinazolinone (2), and 8-hydroxydeoxyvasicinone (3) via novel microwave-assisted domino reactions, as well as a novel…”
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Three-Component One-Pot Total Syntheses of Glyantrypine, Fumiquinazoline F, and Fiscalin B Promoted by Microwave Irradiation by Liu, Ji-Feng, Ye, Ping, Zhang, Bailin, Bi, Grace, Sargent, Katie, Yu, Libing, Yohannes, Daniel, Baldino, Carmen M

“…A microwave-promoted three-component one-pot reaction has been developed to provide access to the core pyrazino[2,1-b]quinazoline-3,6-dione (1) scaffold, which…”
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Microwave-Assisted Concise Total Syntheses of Quinazolinobenzodiazepine Alkaloids by Liu, Ji-Feng, Kaselj, Mira, Isome, Yuko, Chapnick, Jennifer, Zhang, Bailin, Bi, Grace, Yohannes, Daniel, Yu, Libing, Baldino, Carmen M

“…One-pot total syntheses of the quinazolinobenzodiazepine alkaloids sclerotigenin (1), (±)-circumdatin F (2), and (±)-asperlicin C (3) via novel…”
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Microwave-Promoted Suzuki Reactions of Aryl Chlorides in Aqueous Media by Miao, Guobin, Ye, Ping, Yu, Libing, Baldino, Carmen M.

“…The microwave-promoted Suzuki coupling reaction of aryl chlorides with boronic acids performed in an aqueous media was studied using the air- and…”
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Development of α-keto-based inhibitors of cruzain, a cysteine protease implicated in Chagas disease by Choe, Youngchool, Brinen, Linda S., Price, Mark S., Engel, Juan C., Lange, Meinolf, Grisostomi, Corinna, Weston, Scott G., Pallai, Peter V., Cheng, Hong, Hardy, Larry W., Hartsough, David S., McMakin, Marsha, Tilton, Robert F., Baldino, Carmen M., Craik, Charles S.

“…A series of novel α-keto based inhibitors has been developed that covalently binds to the active site of cruzain, a cysteine protease crucial for the life…”
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The accelerated development of an optimized synthesis of 1,2,4-oxadiazoles: application of microwave irradiation and statistical design of experiments by Evans, Marc D, Ring, Jessica, Schoen, Adam, Bell, Andrew, Edwards, Paul, Berthelot, Didier, Nicewonger, Robb, Baldino, Carmen M

“…Herein, we report the development of an optimized microwave-assisted synthesis of 1,2,4-oxadiazoles. The chemistry development process was significantly…”
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Indoloprodigiosins from the C-10 bipyrrolic precursor: New antiproliferative prodigiosin analogs by Baldino, Carmen M., Parr, Jonathan, Wilson, Christopher J., Ng, Shi-Chung, Yohannes, Daniel, Wasserman, Harry H.

“…The condensation of the C-10 methoxybipyrrole precursor ( 3) of prodigiosin with indoles and a related pyrrole derivative yields novel analogs of prodigiosin…”
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Singlet oxygen oxidation of bipyrroles : total synthesis of d,l- and meso-isochrysohermidin by WASSERMAN, H. H, DESIMONE, R. W, BOGER, D. L, BALDINO, C. M

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Access to the noryohimban [6,5,6,5,6] ring system via an intramolecular furan Diels–Alder reaction by Fokas, Demosthenes, Patterson, Jean E., Slobodkin, Gregory, Baldino, Carmen M.

“…Polycyclic indolic compounds containing the [6,5,6,5,6] ring system were prepared via an intramolecular furan Diels–Alder reaction of α,β-unsaturated amides…”
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Incorporation of carbohydrates and peptides into large triazine-based screening libraries using automated parallel synthesis by Gustafson, Gary R., Baldino, Carmen M., O'Donnell, Mary-Margaret E., Sheldon, Adrian, Tarsa, Robert J., Verni, Christopher J., Coffen, David L.

“…A procedure for the sequential, selective derivatization of cyanuric chloride that allows for the incorporation of carbohydrates and peptides has been…”
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Synthesis of 1,2-disubstituted-3-alkylidenylpyrrolidines via a one-pot three-component reaction by Huang, Wenwei, O’Donnell, Mary-Margaret, Bi, Grace, Liu, Jifeng, Yu, Libing, Baldino, Carmen M., Bell, Andrew S., Underwood, Toby J.

“…[Display omitted] Olsson’s three-component reaction of cyclopropylketones, aldehydes, and primary amines was investigated for application to parallel…”
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Selective Oxidation of Phosphorus Ylides by Dimethyldioxirane. Application to the Formation of Vicinal Tricarbonyls by Wasserman, Harry H, Baldino, Carmen M, Coats, Steven J

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Singlet oxygen mediated oxidative decarboxylation of pyrrole-2-carboxylic acids by Boger, Dale L, Baldino, Carmen M

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Singlet Oxygen in Synthesis. Formation of d,l- and meso-Isochrysohermidin from a 3,3′-Bipyrrole Precursor by Wasserman, H

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The synthesis and investigation of the DNA binding properties of dielectrophiles incorporating bis-vicinal tricarbonyls by Wasserman, Harry H., Baldino, Carmen M.

“…A concise and versatile synthesis of bis-vicinal tricarbonyls was developed from readily available diacids or their corresponding diacid chlorides. The…”
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