Search Results - "Atsumi, Eri"

K-685, a TRPV1 Antagonist, Blocks PKC-Sensitized TRPV1 Activation and Improves the Inflammatory Pain in a Rat Complete Freund’s Adjuvant Model by Sugimoto, Yoshiyuki, Kojima, Yozo, Inayoshi, Atsushi, Inoue, Kazuaki, Miura-Kusaka, Hiroko, Mori, Kiyotoshi, Saku, Osamu, Ishida, Hiroshi, Atsumi, Eri, Nakasato, Yoshisuke, Shirakura, Shiro, Toki, Shin-ichiro, Shinoda, Katsumi, Suzuki, Nobuyuki

“…Transient receptor potential vanilloid 1 (TRPV1) is a Ca2+-permeable non-selective cation channel that transmits pain signals. TRPV1 is activated by multiple…”
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Discovery of Novel 5,5-Diarylpentadienamides as Orally Available Transient Receptor Potential Vanilloid 1 (TRPV1) Antagonists by Saku, Osamu, Ishida, Hiroshi, Atsumi, Eri, Sugimoto, Yoshiyuki, Kodaira, Hiroshi, Kato, Yoshimitsu, Shirakura, Shiro, Nakasato, Yoshisuke

“…We have developed a novel and potent chemical series of 5,5-diphenylpentadienamides for targeting TRPV1 in vitro and in vivo. In this investigation, we…”
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