Search Results - "Andrade‐Sampedro, Paula"

Palladium‐Catalyzed Site‐Selective C(sp2)−H Acetoxylation of Tyrosine‐Containing Peptides by Urruzuno, Iñaki, Andrade‐Sampedro, Paula, Correa, Arkaitz

“…A Pd‐catalyzed C(sp2)−H acetoxylation of Tyr‐containing peptides is described. The method relies on the use of a removable 2‐pyridyloxy group as directing…”
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Ru‐Catalyzed C−H Hydroxylation of Tyrosine‐Containing Di‐ and Tripeptides toward the Assembly of L‐DOPA Derivatives by Andrade‐Sampedro, Paula, Matxain, Jon M., Correa, Arkaitz

“…The development of catalytic tools for the late‐stage modification of amino acids within a peptide framework is a challenging task of capital importance…”
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Pd‐Catalyzed C(sp2)−H Alkoxycarbonylation of Phenethyl‐ and Benzylamines with Chloroformates as CO Surrogates by Andrade‐Sampedro, Paula, Matxain, Jon M., Correa, Arkaitz

“…The site‐selective functionalization of C−H bonds within a complex molecule remains a challenging task of capital synthetic importance. Herein, an…”
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On the Mechanism of Cross-Dehydrogenative Couplings between N -aryl Glycinates and Indoles: A Computational Study by Andrade-Sampedro, Paula, Correa, Arkaitz, Matxain, Jon M

“…Despite the widespread use of cross-dehydrogenative couplings in modern organic synthesis, mechanistic studies are still rare in the literature and those…”
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Late-Stage Radical C–H Alkylamination of Tyrosine Compounds and Phenol-Containing Drugs by Andrade-Sampedro, Paula, Correa, Arkaitz

“…A modular site-selective iron-catalyzed radical amination of a number of phenol-containing biomolecules such as tyrosine-containing peptides, estrogens, and…”
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Late-Stage C–H Acylation of Tyrosine-Containing Oligopeptides with Alcohols by Urruzuno, Iñaki, Andrade-Sampedro, Paula, Correa, Arkaitz

“…The selective tagging of amino acids within a peptide framework while using atom-economical C–H counterparts poses an unmet challenge within peptide chemistry…”
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