Search Results - "Adolfsson, Dan E"

Synthesis of Densely Functionalized N‑Alkenyl 2‑Pyridones via Benzyne-Induced Ring Opening of Thiazolino-Fused 2‑Pyridones by Singh, Pardeep, Cairns, Andrew G, Adolfsson, Dan E, Ådén, Jörgen, Sauer, Uwe H, Almqvist, Fredrik

“…We report the synthesis of 6-arylthio-substituted-N-alkenyl 2-pyridones by ring opening of bicyclic thiazolino-2-pyridones with arynes. Varied…”
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Intramolecular Povarov Reactions for the Synthesis of Chromenopyridine Fused 2‑Pyridone Polyheterocycles Binding to α‑Synuclein and Amyloid‑β Fibrils by Adolfsson, Dan E, Tyagi, Mohit, Singh, Pardeep, Deuschmann, Adrian, Ådén, Jörgen, Gharibyan, Anna L, Jayaweera, Sanduni Wasana, Lindgren, Anders E. G, Olofsson, Anders, Almqvist, Fredrik

“…A BF3·OEt2 catalyzed intramolecular Povarov reaction was used to synthesize 15 chromenopyridine fused thiazolino-2-pyridone peptidomimetics. The reaction works…”
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Tandem Ring Opening/Intramolecular [2 + 2] Cycloaddition Reaction for the Synthesis of Cyclobutane Fused Thiazolino-2-Pyridones by Tyagi, Mohit, Adolfsson, Dan E, Singh, Pardeep, Ådén, Jörgen, Jayaweera, Sanduni Wasana, Gharibyan, Anna, Bharate, Jaideep B, Kiss, Anita, Sarkar, Souvik, Olofsson, Anders, Almqvist, Fredrik

“…Reaction of thiazoline fused 2-pyridones with alkyl halides in the presence of cesium carbonate opens the thiazoline ring via S-alkylation and generates…”
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Pyridine-Fused 2‑Pyridones via Povarov and A3 Reactions: Rapid Generation of Highly Functionalized Tricyclic Heterocycles Capable of Amyloid Fibril Binding by Singh, Pardeep, Adolfsson, Dan E, Ådén, Jörgen, Cairns, Andrew G, Bartens, Christian, Brännström, Kristoffer, Olofsson, Anders, Almqvist, Fredrik

“…We here describe the use of three-component reactions to synthesize tricyclic pyridine ring-fused 2-pyridones. The developed protocols have a wide substrate…”
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K 2 S 2 O 8 -mediated coupling of 6-amino-7-aminomethyl-thiazolino-pyridones with aldehydes to construct amyloid affecting pyrimidine-fused thiazolino-2-pyridones by Bharate, Jaideep B, Ådén, Jörgen, Gharibyan, Anna, Adolfsson, Dan E, Jayaweera, Sanduni Wasana, Singh, Pardeep, Vielfort, Katarina, Tyagi, Mohit, Bonde, Mari, Bergström, Sven, Olofsson, Anders, Almqvist, Fredrik

“…We herein present the synthesis of diversely functionalized pyrimidine fused thiazolino-2-pyridones K S O -mediated oxidative coupling of…”
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Pyridine-Fused 2-Pyridones via Povarov and A 3 Reactions: Rapid Generation of Highly Functionalized Tricyclic Heterocycles Capable of Amyloid Fibril Binding by Singh, Pardeep, Adolfsson, Dan E, Ådén, Jörgen, Cairns, Andrew G, Bartens, Christian, Brännström, Kristoffer, Olofsson, Anders, Almqvist, Fredrik

“…We here describe the use of three-component reactions to synthesize tricyclic pyridine ring-fused 2-pyridones. The developed protocols have a wide substrate…”
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