Search Results - "Švarcová, Markéta"
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Substituted N-phenylitaconamides as inhibitors of mycobacteria and mycobacterial isocitrate lyase
Published in European journal of pharmaceutical sciences (01-09-2022)Get full text
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Using historical ecology to reassess the conservation status of coniferous forests in Central Europe
Published in Conservation biology (01-02-2017)“…Forests cover approximately one-third of Central Europe. Oak (Quercus) and European beech (Fagus sylvatica,) are considered the natural dominants at low and…”
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3
Novel Iodinated Hydrazide-hydrazones and their Analogues as Acetyl- and Butyrylcholinesterase Inhibitors
Published in Current topics in medicinal chemistry (01-01-2020)“…Hydrazide-hydrazones have been known as scaffold with various biological activities including inhibition of acetyl- (AChE) and butyrylcholinesterase (BuChE)…”
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New 3-amino-2-thioxothiazolidin-4-one-based inhibitors of acetyl- and butyryl-cholinesterase: synthesis and activity
Published in Future medicinal chemistry (01-01-2024)“…2-Thioxothiazolidin-4-one represents a versatile scaffold in drug development. The authors used it to prepare new potent acetylcholinesterase (AChE) and…”
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Novel Cholinesterase Inhibitors Based on O-Aromatic N,N-Disubstituted Carbamates and Thiocarbamates
Published in Molecules (Basel, Switzerland) (11-02-2016)“…Based on the presence of carbamoyl moiety, twenty salicylanilide N,N-disubstituted (thio)carbamates were investigated using Ellman's method for their ability…”
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N -Alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1-carboxamides and Their Analogues: Synthesis and Multitarget Biological Activity
Published in Molecules (Basel, Switzerland) (12-05-2020)“…Based on the isosterism concept, we have designed and synthesized homologous -alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1-carboxamides (from C to C ) as…”
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Human-induced changes in fire regime and subsequent alteration of the sandstone landscape of Northern Bohemia (Czech Republic)
Published in Holocene (Sevenoaks) (01-03-2018)“…Multiproxy palaeoecological evidence from a sandstone region in northern Czech Republic was collected to explore the impact of fire disturbances on the decline…”
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5-Aryl-1,3,4-oxadiazol-2-amines Decorated with Long Alkyl and Their Analogues: Synthesis, Acetyl- and Butyrylcholinesterase Inhibition and Docking Study
Published in Pharmaceuticals (Basel, Switzerland) (25-03-2022)“…2,5-Disubstituted 1,3,4-oxadiazoles are privileged versatile scaffolds in medicinal chemistry that have exhibited diverse biological activities. Acetyl- (AChE)…”
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Novel Aminoguanidine Hydrazone Analogues: From Potential Antimicrobial Agents to Potent Cholinesterase Inhibitors
Published in Pharmaceuticals (Basel, Switzerland) (26-11-2021)“…A series of thirty-one hydrazones of aminoguanidine, nitroaminoguanidine, 1,3-diaminoguanidine, and (thio)semicarbazide were prepared from various aldehydes,…”
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Divergent fire history trajectories in Central European temperate forests revealed a pronounced influence of broadleaved trees on fire dynamics
Published in Quaternary science reviews (15-10-2019)“…Fire occurrence is driven by a complex interplay between vegetation, climatic, landform and human factors making it challenging to separate the individual…”
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Novel Inhibitors of Acetyl- and Butyrylcholinesterase Derived from Benzohydrazides: Synthesis, Evaluation and Docking Study
Published in Pharmaceuticals (Basel, Switzerland) (24-01-2023)“…On the basis of previous reports, novel 2-benzoylhydrazine-1-carboxamides were designed as potential inhibitors of acetylcholinesterase (AChE) and…”
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Investigation of potential inhibitors of chorismate-utilizing enzymes
Published in Current medicinal chemistry (01-01-2015)“…Chorismate-utilizing enzymes (CUE) such as chorismate mutase, anthranilate synthase, chorismate pyruvate-lyase, 4-amino-4-deoxychorismate synthase,…”
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Změna vnímání genderové rovnosti ve státní správě prostřednictvím nové evropské legislativy?
Published in Gender a výzkum (On-line) (2019)“…V Praze se konal kulatý stůl s názvem „Genderová rovnost a státní správa: Zkušenosti z Evropské komise a OECD“ pořádaný Ministerstvem školství, mládeže a…”
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Historické kořeny problematiky podnikatelek a současná situace podnikatelek v České republice
Published in Gender a výzkum (On-line) (01-12-2018)“…Review of book Ženy-podnikatelky v minulosti a současnosti (Slavíčková P. ed.)…”
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The Sociological Imagination: Do We Build Boundaries or Do We Want Solidarity?
Published in Gender a výzkum (On-line) (01-12-2019)“…Report from the conference Europe and Beyond: Boundaries, Barriers and Belonging…”
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Podnikání matek malých dětí jako prekérní typ zaměstnání? Srovnání zkušeností podnikatelek s malými dětmi původem z ČR a z Ukrajiny
Published in Gender a výzkum (On-line) (01-12-2019)“…Entrepreneurship may be associated with independence and profit, but it may also be a precarious type of employment. Self-employment is often a strategy for…”
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Salicylanilide Diethyl Phosphates as Potential Inhibitors of Some Mycobacterial Enzymes
Published in TheScientificWorld (2014)“…Antimycobacterially active salicylanilide diethyl phosphates were evaluated to identify their potential drug target(s) for the inhibition of several…”
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New lipophilic isoniazid derivatives and their 1,3,4-oxadiazole analogues: Synthesis, antimycobacterial activity and investigation of their mechanism of action
Published in European journal of medicinal chemistry (10-05-2018)“…The development of novel drugs is essential for the treatment of tuberculosis and other mycobacterial infections in future. A series of…”
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